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4-(5-phenyl-1,2-oxazole-4-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
2-methoxyethyl 2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxylate
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-3-phenyl-1H-pyrazole-4-carboxamide
2-{4-[(2,5-dimethoxyphenyl)methyl]-1-(2,2-dimethylpropyl)piperazin-2-yl}ethan-1-ol
(4aS,8aR)-6-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
4-[(3S)-3-aminopyrrolidine-1-carbonyl]-N-[3-(propan-2-yloxy)propyl]benzene-1-sulfonamide
4-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]piperazine-1-carboxamide
(3R,4R)-1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
2-(3-{[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]methyl}-1H-indol-1-yl)acetamide
4-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
3-(4-methyl-1,3-thiazol-5-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]propanamide
1-[3-oxo-3-(pyrrolidin-1-yl)propyl]-3-propylpiperidine-3-carboxylic acid
N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-4-sulfamoylbenzamide
4-(2-methoxyphenoxy)-1-[(trimethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylic acid
N-(3-{4-[4-(2-hydroxyphenyl)piperazin-1-yl]piperidin-1-yl}phenyl)-4-phenylbutanamide
ethyl 5-(1H-imidazol-2-ylmethyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-[(4-fluorophenyl)methyl]-1-[(2-methoxypyrimidin-5-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-(cyclopropylmethyl)-N-propyl-3-(1H-1,2,3,4-tetrazol-1-yl)-5-(2,3,4-trimethoxyphenyl)benzamide
4-oxo-1-[(2S)-oxolan-2-ylmethyl]-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-N-(5,6,7,8-tetrahydronaphthalen-1-yl)benzamide
3-{2-[4-(furan-3-carbonyl)-1,4-diazepan-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
methyl 5-oxo-5-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]pentanoate
3-hydroxy-1-(2-phenylethyl)-3-{[(2-phenylpropan-2-yl)amino]methyl}piperidin-2-one
ethyl 5-{2-azabicyclo[2.2.1]heptan-2-ylmethyl}-1-(4-methoxyphenyl)-1H-pyrazole-4-carboxylate
4-methyl-2-(2-{2-[1-(propan-2-yl)piperidin-4-yl]acetamido}ethyl)-1,3-thiazole-5-carboxylic acid
1-(4-{4-[(oxan-3-ylmethyl)amino]piperidin-1-yl}phenyl)pyrrolidin-2-one
1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
4-({4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)-1-methyl-1H-pyrrole-2-carbonitrile
N-(1-carbamoylcyclopentyl)-5-(methoxymethyl)furan-2-carboxamide
N-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
1-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-2-methylpropan-1-one
N2-[1-(4-fluorophenyl)pyrrolidin-3-yl]-N1-(pyridin-3-yl)ethane-1,2-diamine
3-(3-chloro-4-propoxyphenyl)-1-[1-(pyridin-3-yl)propyl]urea
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-2,6,8-trimethylquinoline-4-carboxamide
{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}(thiophen-2-yl)methanol
(1R,5R)-6-[2-(benzenesulfonyl)ethyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-methyl-2-[methyl(1-methylpiperidin-4-yl)amino]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-3,4-dimethylbenzamide
N-[(3R,4S)-4-cyclopropyl-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}pyrrolidin-3-yl]-2-hydroxyacetamide
1-{2-[methyl(oxolan-2-ylmethyl)amino]pyrimidin-4-yl}piperidin-4-ol
4-methoxy-2-{4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}phenol
1-(5-{[(dicyclopropylmethyl)amino]methyl}-2-methoxyphenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
1-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-(1H-1,2,3,4-tetrazol-5-yl)ethan-1-one
2-{3-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-1H-pyrazol-1-yl}-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(6-methylpyridin-2-yl)methyl]acetamide
{[4-(butan-2-yloxy)-3-chlorophenyl]methyl}[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]amine
N,1-dimethyl-4-oxo-N-[1-(pyridin-3-yl)propyl]-1,4-dihydroquinoline-3-carboxamide
(3aR,6aS)-5-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-2-ethyl-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(2-fluorophenyl)methyl]-N-(2-hydroxyethyl)-6-oxopiperidine-3-carboxamide
3-chloro-2-(2,5-dimethoxyphenyl)-5-methylpyridine