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N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(pyridin-2-ylmethyl)piperidin-4-amine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methyl-1,3-oxazole-4-carboxamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}methanesulfonamide
7-(2-methoxyethyl)-2-(8-methoxyquinolin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-4-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
2-{[2-(pyridin-3-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
3-(5-methylfuran-2-yl)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-1H-pyrazole-5-carboxamide
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4-(2-methylpyridin-4-yl)piperazine
methyl 3-cyclohexaneamido-6-(morpholin-4-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-{4-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenyl}acetamide
4-(4-methyl-1H-pyrazol-1-yl)-1-[3-(5-methylfuran-2-yl)butyl]piperidine-4-carboxylic acid
2-(3-fluoro-4-hydroxyphenyl)-1-[3-(pyridin-3-yl)azetidin-1-yl]ethan-1-one
3-methyl-1-[2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidin-3-ol
7-[(3-methoxyphenyl)methyl]-2-(oxane-4-carbonyl)-2,7-diazaspiro[4.5]decane
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
1,6-dimethyl-N-{1-oxaspiro[4.5]decan-3-yl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(6-hydroxy-4-{thieno[3,2-d]pyrimidin-4-yl}-1,4-diazepan-1-yl)ethan-1-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(2,6-difluorophenyl)methyl]benzamide
1-[2-(ethylsulfanyl)-1,3-benzoxazol-6-yl]-3-methyl-3-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea
4-{2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-2-methoxypyridine-3-carbonitrile
6-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N-{2-[5-methyl-4-({methyl[(1-phenyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1,3-oxazol-2-yl]phenyl}thiophene-3-carboxamide
1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
3-methoxy-1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
2-(2-methoxyethyl)-8-(4-oxo-4-phenylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
1,3-dimethyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-1H-indole-2-carboxamide
N-(2-ethoxyphenyl)-3-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]-3-oxopropanamide
3-(1-{1-[2-(diethylamino)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(3-fluorophenyl)urea
2-[5-(1-benzofuran-2-yl)-4-phenyl-1H-imidazol-1-yl]-1-(pyridin-3-yl)ethan-1-ol
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
6-(benzyloxy)-1-cyclohexyl-4-(oxolane-3-carbonyl)-1,4-diazepan-2-one
4-(2,5-dimethoxyphenyl)-2-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)phenol
5-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-({1-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetyl]piperidin-3-yl}methyl)furan-2-carboxamide
4-phenyl-1-(3-phenylpropyl)-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-phenyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1,2-oxazole-3-carboxamide
(2S)-N1-(2-methoxyethyl)-N2-[3-(3-methylphenyl)phenyl]pyrrolidine-1,2-dicarboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]ethan-1-one
7-fluoro-N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-methylquinoline-4-carboxamide
N-(3-hydroxypropyl)-2-(2-oxopyrrolidin-1-yl)-N-(pyridin-4-ylmethyl)propanamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
3-methyl-3-[(4-methyl-1H-imidazol-2-yl)methyl]-1-[2-(morpholin-4-ylmethyl)phenyl]urea
N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
2-(2-{[(2,2-dimethylcyclopropyl)methyl](methyl)amino}-4-(morpholin-4-yl)pyrimidin-5-yl)-2-methylpropanoic acid
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-(1-ethyl-1H-indole-5-carbonyl)-1-(4-methylphenyl)piperazin-2-one
8-[4-(difluoromethoxy)benzoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-{5-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid