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6-{4-[(3-methoxypropyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}-2,3-dihydropyridazin-3-one
2-(1-tert-butyl-1H-pyrrole-3-carbonyl)-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
3,5-dimethyl-2-[2-(morpholin-4-ylmethyl)-1,4-oxazepane-4-carbonyl]-1H-indole
1-[2-(1H-imidazol-2-yl)benzoyl]-2-[2-(thiophen-2-yl)ethyl]piperidine
2-(2-methyl-1H-indol-3-yl)-N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}acetamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-N,N-dimethylpiperidine-1-sulfonamide
1-(1,2,3,4-tetrahydroisoquinolin-2-yl)-3-[2-(thiomorpholin-4-ylmethyl)phenoxy]propan-2-ol
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)acetamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
2-[4-(4-ethyl-2,5-dioxoimidazolidin-4-yl)piperidin-1-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
2,5-dimethyl-N-({5-methyl-2-[2-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)furan-3-carboxamide
1-{[1-(2-hydroxybutyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-2-methyl-1,4-dihydroquinolin-4-one
2-amino-4-{methyl[2-(1H-pyrazol-4-yl)ethyl]amino}quinazoline-6-carboxylic acid
4-[5-(1H-pyrazol-3-yl)furan-2-yl]-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-methyl-6-{5-[1-(1H-pyrazol-1-yl)propyl]-1,2,4-oxadiazol-3-yl}pyridazine
1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
2-[(3,4-difluorophenyl)methyl]-8-(1H-imidazol-4-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-methyl-1H-1,3-benzodiazole
5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylpropanamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazole-3-carboxamide
3-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-5-chloro-1,2-dihydropyridin-2-one
3-(1-{2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-imidazol-2-yl)benzonitrile
2-{2-chloro-6-methoxy-4-[(2-methyl-5-oxo-1,4-diazepan-1-yl)methyl]phenoxy}acetamide
4-[3-(benzyloxy)propyl]-1-(3-methoxyphenyl)piperazin-2-one
7-methyl-2-[2-(methylsulfanyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-[2-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)phenyl]ethan-1-one
3-(2-amino-1,3-thiazol-4-yl)-1-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}propan-1-one
2-{1-cyclopentyl-4-[(3-ethoxy-4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-(furan-2-ylmethyl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
1-[2-({[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}(methyl)amino)ethyl]piperidin-2-one
1-methyl-N,N-bis(1,3-oxazol-4-ylmethyl)-2-oxo-1,2-dihydroquinoline-3-carboxamide
3-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-1-[(1-methyl-1H-imidazol-2-yl)(phenyl)methyl]urea
2-({4-[1-(2-hydroxyethyl)-3-methyl-1H-1,2,4-triazol-5-yl]phenyl}(methyl)amino)ethan-1-ol
3-{5-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-5-(pyrrolidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole
4-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[(2R)-2-hydroxypropyl]-3-methoxybenzamide
1-[(2R)-2-amino-4-methylpentanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-fluoro-N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-5-sulfamoylbenzamide
N,2-dimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
N-(1-benzyl-1H-pyrazol-5-yl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carboxamide
6-cyclobutyl-2-{3-[(3-hydroxyazetidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-{[(1,3-thiazol-2-yl)carbamoyl]methyl}propanamide
1-(cyclopropylmethyl)-6-(dimethyl-1,3-thiazole-5-carbonyl)-3-(2-methylquinolin-5-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-methyl-6-(2-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)pyrimidin-4-ol
(3S,4R)-3-benzyl-1-(3,6-dimethylpyrazin-2-yl)-4-methylpiperidin-4-ol
9-{1-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]piperidin-4-yl}-6-oxa-9-azaspiro[4.5]decane
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-3-ethyl-5-methyl-1,2-oxazole-4-carboxamide
2-({[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(benzyl)amino)ethan-1-ol
1-benzyl-N-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-amine