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2-(2-methylpropyl)-N-[4-(1,3-thiazol-4-yl)phenyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
4-methyl-2-{[3-(3-{pyrazolo[1,5-a]pyrimidin-3-yl}phenyl)-1H-pyrazol-1-yl]methyl}-1,3-thiazole
7-chloro-2-{[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
1-[(3-fluorophenyl)methyl]-4-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
2-(4-methyl-6-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}pyrimidin-2-yl)phenol
2-(4-fluoro-3-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)acetic acid
N-[(2,4-dimethoxyphenyl)methyl]-5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethylpyrazolo[1,5-a]pyridine-3-carboxamide
5-[(3-methoxyphenyl)methyl]-N,N-dimethyl-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-(2-{[3-(dimethylsulfamoyl)-5-{[(4-methylphenyl)methyl]amino}phenyl]formamido}ethyl)acetamide
N-methyl-5-{[5-oxo-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]methyl}furan-2-carboxamide
4-(5-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)pyridine
1-(4-{[3-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,2-oxazol-5-yl]methoxy}phenyl)ethan-1-one
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N,3,5,7-tetramethyl-1H-indole-2-carboxamide
N-(1-ethyl-2-methyl-1H-indol-5-yl)-4-methyl-1,4-diazepane-1-carboxamide
7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-[5-(4-methoxyphenyl)furan-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
4-phenoxy-1-[2-(pyridin-4-yl)acetyl]piperidine-4-carboxylic acid
5-chloro-2-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2,3-dihydro-1H-indole
4-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
1-cyclohexyl-3-(cyclopropylmethyl)-5-[4-(methylamino)piperidine-1-carbonyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-({3-[(2,2-difluoroacetamido)methyl]piperidin-1-yl}methyl)benzoic acid
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(3-methoxypropyl)-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]acetamide
1-acetyl-N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}piperidine-4-carboxamide
6-[4-(4-fluorophenyl)benzoyl]-1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane
2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-6-(4-methylpiperazine-1-carbonyl)pyrazine
(2S)-2-amino-N-[(1-benzylpiperidin-4-yl)methyl]-2-cyclohexyl-N-methylacetamide
4-ethyl-3-[1-(6-phenylpyridazin-3-yl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-(dimethylamino)-2-(4-methylphenyl)ethan-1-one
1-ethyl-N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}-3,5-dimethyl-1H-pyrazole-4-carboxamide
2-{[4-(furan-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-4-(propan-2-yl)-1,3-thiazole
4-[5-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)thiophen-2-yl]-2-methylbut-3-yn-2-ol
4-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methoxypyrimidine
[(3R,4R)-1-(5-ethyl-1,3,4-thiadiazol-2-yl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
4-cyclopentyl-3-{2-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}piperazin-2-one
1-(2,3-dihydro-1H-indol-1-yl)-2-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-methyl-4-(3-{1-[(4-methyl-1,3-thiazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
4-[(6-hydroxy-1,4-oxazepan-6-yl)methyl]-1-(2-phenylethyl)piperazin-2-one
2-butyl-8-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-methoxy-N-methylacetamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
1-{4-[5-(3,4-dimethylpiperazine-1-carbonyl)-2-methoxyphenoxy]piperidin-1-yl}ethan-1-one
3-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-[4-(propan-2-yl)phenyl]urea
methyl 3-(oxolane-3-amido)-1-(3-phenylpropyl)-5-[(4,4,4-trifluorobutan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(5-fluoro-1H-indol-2-yl)methyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
N,2-dimethyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-{3-[4-(oxolane-2-carbonyl)-1,4-diazepan-1-yl]propanamido}benzamide
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine