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2-(2-methylphenyl)-5-{[4-(pyrazin-2-yl)piperazin-1-yl]methyl}pyrimidine
7-[(3-methoxyphenyl)methyl]-2-(2-methylpyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2,4-dimethoxybenzamide
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
1-(cyclohexylmethyl)-3-hydroxy-3-{[4-(propan-2-yl)piperazin-1-yl]methyl}piperidin-2-one
4-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1-[(3-fluorophenyl)methyl]piperazin-2-one
ethyl 1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
2-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}-2-[3-(methylsulfanyl)phenyl]acetic acid
2-ethyl-6-methyl-5-{2-oxo-2-[4-(pyridin-3-yloxy)piperidin-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
(3R,4R)-4-amino-1-(3-chloro-4-methoxybenzoyl)piperidin-3-ol
(4-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}morpholin-2-yl)methanamine
3-amino-1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-hydroxybenzamide
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-3-(2-fluorophenyl)propan-1-one
(2-{1-[(3-fluoro-4-methoxyphenyl)methyl]piperidin-2-yl}ethyl)dimethylamine
10-methoxy-5-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
4-[(1-methoxybutan-2-yl)amino]-5-methyl-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
4-chloro-3-({ethyl[(1-ethyl-1H-pyrazol-4-yl)methyl]carbamoyl}amino)-N-methylbenzamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-(2-methyl-4-phenylpyridine-3-carbonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}-1-(propan-2-yl)-1H-1,3-benzodiazole
(1S,3R)-3-[3-(4-methyl-1,3-thiazol-5-yl)propanamido]-N-phenylcyclopentane-1-carboxamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-(1-methyl-1H-pyrazol-4-yl)-2-{4-[1-(3-methylpyridin-2-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}acetamide
1-(2-methoxyphenyl)-4-{[2-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-one
(4-{2-methylthieno[2,3-d]pyrimidin-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
N-(3,4-dimethylphenyl)-4-[5-(4-methoxybenzamido)-1H-pyrazol-1-yl]piperidine-1-carboxamide
7-[(2-fluoro-4-methoxyphenyl)methyl]-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
4-(2-chlorophenoxy)-1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
N-(2-methylpropyl)-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-4-phenoxybutan-1-one
3-(2-ethyl-1H-imidazol-1-yl)-1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)propan-1-one
1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]urea
6-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
(1S,5R)-6-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
1-methanesulfonyl-4-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-1,4-diazepane
6-(3-carbamoylpiperidin-1-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-[(8-methoxyquinolin-5-yl)methyl]-1-methylurea
(3S,4S)-1-(3-methoxypyridine-2-carbonyl)-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
methyl 5-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
N-[3-hydroxy-1-(4-methylphenyl)propyl]-4-(1H-pyrazol-3-yl)benzamide
(3R,4R)-4-amino-1-({4-amino-6-[(3-methylphenyl)amino]-1,3,5-triazin-2-yl}methyl)piperidin-3-ol
N-(2-methylphenyl)-3-[(3S,4R)-1-(pyridin-2-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
3-hydroxy-1-(2-methoxyethyl)-3-{[4-(propan-2-yl)piperidin-1-yl]methyl}piperidin-2-one
N-(1,3-dihydro-2-benzofuran-5-yl)-3-(pyrimidin-4-yl)piperidine-1-carboxamide
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(1-methylpiperidine-3-carbonyl)piperidine
3-methyl-3-phenyl-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
2-(1H-1,3-benzodiazol-1-yl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}propanamide
2-(cyclopentylmethyl)-6-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-4-oxo-1-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide