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N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-2,5-dihydro-1H-pyrrole-2-carboxamide
2-(propylsulfanyl)-5-{[3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl}pyrimidine
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(oxolane-3-carbonyl)piperidine-4-carboxamide
1-(oxolan-3-ylmethyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-({1-[2-(pyridin-3-yl)acetyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
(3S,4R)-3-methoxy-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-4-amine
(1-{4-[(2-methoxyethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carbonyl}piperidin-2-yl)methanol
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-(4-methylphthalazin-1-yl)pyrrolidin-3-yl]methanol
4-(3-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}phenyl)phenol
ethyl 1-[(2-ethylphenyl)carbamoyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
N-[(3-methoxyphenyl)methyl]-1-methyl-N-(prop-2-en-1-yl)-1H-pyrrole-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopentyl-1-phenyl-1H-1,2,3-triazole-4-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-(pyrrolidin-1-yl)pyridine-3-carboxamide
1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-4-[3-(trifluoromethyl)phenoxy]piperidine
4-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-(3-methoxyphenyl)piperazin-2-one
[(3R,4R)-4-[(dimethylamino)methyl]-1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]methanol
2-(2-methylpropyl)-4-[5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carbonyl]morpholine
2-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
N-(oxolan-3-yl)-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
3-hydroxy-1-{6-hydroxy-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-1,4-diazepan-1-yl}propan-1-one
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]propanamide
5-[(3-methoxyphenyl)methyl]-5-{3-oxo-3-[4-(quinazolin-2-yl)piperazin-1-yl]propyl}pyrrolidin-2-one
4-{5-[3-(3-ethylphenoxy)azetidine-1-carbonyl]pyrimidin-2-yl}morpholine
5-[2-(3-chlorophenoxy)propanoyl]-1-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(cyclohex-1-en-1-ylmethyl)-1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-amine
N-[(2,4-dimethoxyphenyl)methyl]-3-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)propanamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-(propan-2-yl)acetamide
4-{[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]sulfonyl}morpholine
methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})(pyridin-3-ylmethyl)amine
8-fluoro-4-oxo-N-[3-(propan-2-yloxy)propyl]-1,4-dihydroquinoline-2-carboxamide
methyl({[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})(propan-2-yl)amine
2-(2-hydroxyethyl)-8-[2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
5-(2-fluorophenyl)-N-(1H-imidazol-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
1-{4-[(cyclopentylamino)methyl]-2-methoxyphenoxy}-3-(4-ethylpiperazin-1-yl)propan-2-ol
(1S,5R)-6-(2,4-dimethoxybenzoyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-{3-methyl-5-[2-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
2-(1,4-dimethylpiperazin-2-yl)-N-{[(2-methylphenyl)carbamoyl]methyl}acetamide
N-(2-methoxyethyl)-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
8-[4-(1H-imidazol-1-yl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
7-(3-chlorophenyl)-4-cyclopentanecarbonyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(1-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)-N-cyclopropylpropanamide
1-[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]-3-[2-(N-methylmethanesulfonamido)ethyl]urea
2-[(4-{2-ethyl-3H-imidazo[4,5-b]pyridin-6-yl}-1H-pyrrolo[2,3-b]pyridin-6-yl)amino]ethan-1-ol
2-(dimethylamino)-2-(4-fluorophenyl)-N-(oxan-4-yl)acetamide
2-(1H-indazol-3-yl)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
1-methyl-2-(2-methylpyrimidin-5-yl)-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazole
(1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)methanamine