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N-benzyl-4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
2-benzyl-9-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(cyclohex-1-en-1-yl)ethyl]-5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)pyrrolidin-2-one
[4-(2,3-dihydro-1,4-benzodioxin-6-yl)pyridin-2-yl]methanol
N-[1-(cyclopropylmethyl)-1H-indazol-3-yl]-2-[3-(thiophen-3-yl)-1H-pyrazol-1-yl]acetamide
5-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1-(2-methylpropyl)piperidin-2-one
(1S,5R)-6-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
N-ethyl-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]-N-(2,2,2-trifluoroethyl)acetamide
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-3-phenylpiperazine
3-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-2H-indazole
2-amino-6-(5-methylfuran-2-yl)-4-[3-(morpholin-4-ylmethyl)phenyl]pyridine-3-carbonitrile
4-(1,2-oxazolidine-2-carbonyl)-N-propylbenzene-1-sulfonamide
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(4-methyl-1H-imidazole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
7,7-dimethyl-2-[(1-methylpiperidin-4-yl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-methyl-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-(quinoxalin-2-ylmethyl)acetamide
4-[(1-methyl-1H-imidazol-5-yl)methyl]-2-(morpholin-4-ylmethyl)-1,4-oxazepane
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(oxan-4-ylmethyl)amine
2-amino-4-[4-(3-hydroxyprop-1-yn-1-yl)phenyl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
N-(2,1,3-benzothiadiazol-5-ylmethyl)-7-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
6-methyl-2-[3-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile
6-fluoro-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
methyl 4-[4-(2-chloro-4-{[2-(dimethylamino)ethyl]carbamoyl}phenoxy)piperidin-1-yl]-4-oxobutanoate
3-{3-methyl-5-[2-(2-methyl-1H-indol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
2-(2-methoxyethyl)-6-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}-1,3-benzoxazole
5-[3-(2-fluorophenyl)-1H-pyrazol-4-yl]-3-(oxolan-2-ylmethyl)-1,2,4-oxadiazole
N-[2-(2-oxopiperidin-1-yl)ethyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
1,4-dimethyl-9-{[1-(4-methylpyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,4,9-triazaspiro[5.5]undecane
(5S,9aS,9bS)-5-(2-methoxyphenyl)-2-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
7-methoxy-2-[4-(3-methoxypropyl)piperazin-1-yl]-4-methylquinazoline
N-[(2-ethoxyphenyl)methyl]quinoxalin-6-amine
4-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-2-fluorophenol
3-({2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]pyrimidin-4-yl}(methyl)amino)propane-1,2-diol
1-(1H-pyrrole-2-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
4-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}phenol
7-(2-methoxyethoxy)-4-[3-(1H-pyrazol-1-yl)phenyl]-1,2,3,4-tetrahydroquinolin-2-one
2-methyl-6-(1-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)pyrimidin-4-ol
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-[(pyridin-3-ylmethyl)amino]pyridine-3-carboxamide
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
2-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-N,N-dimethylacetamide
3-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1-[4-(trifluoromethoxy)phenyl]urea
2-[1-(4-chlorophenyl)-3-(furan-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-[(2R)-2-hydroxypropyl]acetamide
1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-3,4,4-trimethylpyrrolidin-3-ol
2-[1-(4-propoxybenzoyl)azetidin-3-yl]pyridine
benzyl(cyclopropylmethyl){[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}amine
5-(methoxymethyl)-N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)furan-2-carboxamide
6-{spiro[indene-1,4'-piperidine]-1'-ylmethyl}-1,4-oxazepan-6-ol
[(3R,4R)-1-(2H-1,3-benzodioxole-5-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-(2-ethoxyethyl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(methoxymethyl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-(pyridine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide