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5-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2-methyl-1,3-benzothiazole
2-amino-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-6-(propan-2-yl)pyrimidine-4-carboxamide
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)cyclohexanecarboxamide
5-[3-(3-methylphenyl)-1H-pyrazol-4-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-[3-(difluoromethyl)-5-methyl-1H-pyrazol-1-yl]-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]acetamide
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(propan-2-yloxy)ethan-1-one
2-chloro-4-({[2-(morpholin-4-yl)ethyl]carbamoyl}amino)-N-(propan-2-yl)benzamide
(3S,5R,9R)-5-hydroxy-11-(naphthalene-2-carbonyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
N-{1-[1-(propan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
3-methyl-5-{pyrazolo[1,5-a]pyridin-7-yl}pyridin-2-amine
3-fluoro-2-methoxy-N-methyl-N-[(5-methylfuran-2-yl)methyl]benzamide
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]({[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl})amine
3-(2-methoxyethyl)-3-[(5-methylthiophen-2-yl)methyl]-1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
6-(methoxymethyl)-1-methyl-N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-(2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N3-cyclooctyl-N5-[(1-hydroxycyclohexyl)methyl]-1-(2-methoxyethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-benzyl-5-(4-ethylpiperazin-1-yl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
6-[3-(1H-imidazol-1-yl)propyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-(4-phenoxybenzoyl)-1-(propane-2-sulfonyl)piperidine
N-(adamantan-1-ylmethyl)-N-(2-hydroxyethyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N,N-bis(prop-2-en-1-yl)propanamide
2-(4-fluorophenyl)-N-(2-{7-[(2-hydroxy-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
methyl 1-(2-methoxyethyl)-5-{[(4-methoxyphenyl)methyl]amino}-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidin-3-yl]methanol
1-{1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]piperidin-4-yl}pyrrolidin-2-one
6-(aminomethyl)-N-[2-(2-fluorophenoxy)ethyl]pyrimidin-4-amine
N,N-dimethyl-3-({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}sulfamoyl)benzamide
diethyl({3-[4-(2-methoxyethyl)piperazine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-[(6-methylpyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
(1S,2R)-1-{[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]amino}-2,3-dihydro-1H-inden-2-ol
2-(cyclopropylmethyl)-9-(4-hydroxybenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl({2-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl})(thiophen-2-ylmethyl)amine
N-[2-(1,3-benzothiazol-2-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-[6-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]propan-1-ol
2-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-3-(piperidine-1-carbonyl)pyrazine
4-(4-methoxyphenoxy)-1-(oxolane-3-carbonyl)piperidine
N-{2-[(3S,4S)-3,4-dihydroxypiperidine-1-carbonyl]phenyl}-5-(methoxymethyl)furan-2-carboxamide
3-(4-methylphenyl)-N-[2-(oxolane-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]propanamide
1-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
2-methyl-6-(propan-2-yl)-N-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]pyrimidin-4-amine
2-(4-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperazin-1-yl)pyridine-3-carbonitrile
1-[2-({[4-(furan-2-yl)phenyl]carbamoyl}amino)ethyl]piperidine-3-carboxamide
methyl (1R,3S,3aR,6aS)-3-[4-hydroxy-3-methoxy-5-(prop-2-en-1-yl)phenyl]-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
6-{[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}pyridine-2-carboxylic acid
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(pyrrolidin-1-yl)benzamide
(1S,5R)-3-cycloheptyl-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl (1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
N-(2-methoxyethyl)-6-(4-methoxyphenyl)-N,7-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[1-({[2-(furan-2-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-phenoxyacetamide
6-(2,5-dimethylphenyl)-N,N-dimethylpyridine-2-carboxamide