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1-methyl-4-{4-[4-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]phenyl}piperazine
2-amino-7-hydroxy-4-[5-(hydroxymethyl)furan-2-yl]-5H-indeno[1,2-b]pyridine-3-carbonitrile
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
(2S,4S)-N,N-diethyl-4-[2-(1H-indol-1-yl)acetamido]-1-methylpyrrolidine-2-carboxamide
2-[2-({1-[3-(3-methylphenyl)phenyl]piperidin-4-yl}amino)ethoxy]ethan-1-ol
N-methyl-1-(piperidin-3-ylmethyl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-{6-methoxy-2-oxo-4-[2-(propan-2-yl)pyrimidin-4-yl]-1,2,3,4-tetrahydroquinolin-7-yl}propanamide
{3-[(3-chlorophenyl)methyl]-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-3-yl}methanol
1-{6-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]pyrimidin-4-yl}piperidin-4-ol
2-ethyl-9-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecane
3-{2-[2-(cyclohexylmethyl)morpholin-4-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
3-chloro-4-fluoro-N-[2-(1H-pyrazol-4-yl)ethyl]-1-benzothiophene-2-carboxamide
(3S,4S)-1-{4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carbonyl}-4-(propan-2-yloxy)pyrrolidin-3-ol
1-[2-(2,4-dimethylphenoxy)ethyl]-4-ethyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 3-[(3S,4R)-1-(1H-indol-3-ylmethyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoate
(4-{[(6-cyclopropylpyrimidin-4-yl)(methyl)amino]methyl}oxan-4-yl)methanol
1-(4-ethoxy-2-fluorophenyl)-3-[3-(methylsulfanyl)propyl]urea
N-[2-(but-3-enoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-(4-methylphenyl)propanamide
7-[(4-fluorophenyl)methyl]-2-(pyridine-3-sulfonyl)-2,7-diazaspiro[4.5]decane
2,3,4-trifluoro-N-methyl-N-(quinolin-5-ylmethyl)benzamide
4-[2,5-dichloro-4-(1H-pyrrol-1-yl)phenyl]-4H-1,2,4-triazole
3-{2-[4-(1-hydroxypropyl)piperidin-1-yl]-2-oxoethyl}-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidine-2,5-dione
N-methyl-2-(1H-pyrazol-1-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}butanamide
N-cyclohexyl-N-(2-hydroxy-2-phenylethyl)-3-(1-methyl-1H-pyrazol-5-yl)propanamide
1,9-dimethyl-4-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N5-(butan-2-yl)-1-cyclopentyl-4-oxo-N3,N3-bis(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
5-(4-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}phenyl)-2H-1,2,3,4-tetrazole
1-(4-{[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
methyl 2-{N-methyl-1-[6-oxo-1-(2-phenylethyl)piperidin-3-yl]formamido}acetate
4-(dimethyl-1,2-oxazole-4-carbonyl)-1-phenylpiperazin-2-one
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidine-2-carboxylic acid
1-{[2-(pyridin-2-yl)piperidin-1-yl]sulfonyl}azepane
(1S,6R)-9-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
3-cyclopropyl-5-(furan-2-yl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-ethyl-N-[2-(phenylsulfanyl)ethyl]acetamide
methyl 3-[(2S)-1-acetylpyrrolidine-2-carbonyl]-9-(cyclopentyloxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[(6-methylpyridin-2-yl)methyl]acetamide
1-[2-(cyclobutylformamido)ethyl]-N-(2-methylphenyl)-1H-1,2,3-triazole-4-carboxamide
3-{[3-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}benzoic acid
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-methyl-1-(2-phenylethyl)piperidin-3-amine
6-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-(cyclohexylmethyl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
5-ethyl-N-[2-(1H-imidazol-1-yl)ethyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-(2-hydroxyethyl)-N-(2-methoxy-5-phenylphenyl)-3-oxopiperazine-1-carboxamide
1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[(3-methylphenyl)sulfanyl]piperidine
(2S,4R)-1-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-N-ethyl-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
N-benzyl-1-(1-propanoylpiperidin-4-yl)piperidine-3-carboxamide
3-oxo-N-(5-oxo-1-propylpyrrolidin-3-yl)-3,4-dihydroquinoxaline-2-carboxamide
2-(2,5-dimethylphenoxy)-N-(2-methanesulfonylethyl)propanamide
3-[5-(2-phenylethyl)-1,3,4-thiadiazol-2-yl]-1-[2-(pyrrolidin-1-yl)ethyl]urea