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N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}morpholine-4-sulfonamide
N-[(3R,4S)-4-cyclopropyl-1-(4,4,4-trifluorobutanoyl)pyrrolidin-3-yl]methanesulfonamide
1-amino-N-{[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-4-yl]methyl}cyclopropane-1-carboxamide
N-[2-(dimethylsulfamoyl)ethyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
4-(cyclopropylmethyl)-9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl 1-({4-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
1-[(1-ethyl-1H-imidazol-5-yl)methyl]-4-(5-ethylfuran-2-yl)-1H-1,2,3-triazole
3-{1-[6-(dimethylamino)pyridine-3-carbonyl]piperidin-4-yl}phenol
N,N-dimethyl-3-({3-oxo-2-azaspiro[4.5]decan-2-yl}methyl)-1,2,4-oxadiazole-5-carboxamide
1-({1-[(2-methoxypyrimidin-5-yl)methyl]pyrrolidin-3-yl}methyl)-3-(propan-2-yl)urea
(2S,4R)-N-ethyl-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[2-(thiophen-2-yl)acetamido]pyrrolidine-2-carboxamide
N-(1-{2-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-(phenylsulfanyl)acetamide
4-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-2-amine
6-ethyl-2-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)quinoline-4-carboxamide
9-(furan-3-ylmethyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-methyl-1-(prop-2-en-1-yl)-3-({[2-(pyridin-2-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
2-[4-(propan-2-yl)morpholin-2-yl]-N-{[2-(trifluoromethyl)phenyl]methyl}acetamide
(4S)-1-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3,3,4-trimethylpiperidin-4-ol
N-(3,4-difluorophenyl)-1-[(3,4-dimethoxyphenyl)methyl]piperidin-3-amine
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]acetamide
N-methyl-3-[1-(2-methylpyrimidine-5-carbonyl)piperidin-3-yl]-N-[2-(pyridin-2-yl)ethyl]propanamide
N-(cyclopropylmethyl)-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-(oxolan-2-ylmethyl)acetamide
4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-[(2E)-2-methylbut-2-en-1-yl]piperidine
3-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-1-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}urea
2-(3,5-dimethylphenyl)-2-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidin-1-yl}acetic acid
7-fluoro-3-{2-[1-(propan-2-yl)piperidin-2-yl]ethyl}-3,4-dihydroquinazolin-4-one
(1R,5R)-6-methyl-3-(5-methylthiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
{[7-methoxy-2-(thiophen-2-yl)quinolin-3-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
3-(1-{3-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]propanoyl}piperidin-4-yl)-N-phenylpropanamide
9-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-6-oxa-9-azaspiro[4.5]decane
methyl 3-({imidazo[1,2-a]pyridin-2-ylformamido}methyl)-5-(thiophene-2-sulfonamido)benzoate
2-(2,2-dimethylpropanamido)-5-methyl-N-[3-(pyridin-4-yl)propyl]thiophene-3-carboxamide
N-(1-{7-[(4-methoxy-2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
(3S,4S)-1-(1,3-benzothiazol-2-yl)-4-(morpholin-4-yl)pyrrolidin-3-ol
3-[(5-fluoro-1H-indol-2-yl)methyl]-3H,4H-pyrido[3,4-d]pyrimidin-4-one
3,4-difluoro-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)benzamide
4-methyl-2-[4-(2-methyloxolane-2-carbonyl)piperazin-1-yl]-6-(trifluoromethyl)pyrimidine
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-amino-4-(1-ethyl-1H-pyrazol-4-yl)-6-(thiophene-2-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
2-(3-methoxyphenyl)-1-[5-(4-methoxyphenyl)furan-2-carbonyl]azetidine
{1-[2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidin-3-yl}methanol
4-[(2-butyl-1H-imidazol-4-yl)methyl]-7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-(2-chloro-4-methoxyphenoxymethyl)-N-[(1r,4r)-4-hydroxycyclohexyl]-1H-pyrazole-3-carboxamide
4-(2,3-dihydroxybenzoyl)-1-(4-methylphenyl)piperazin-2-one
3,4,7-trimethyl-2-[3-(propoxymethyl)pyrrolidine-1-carbonyl]-1H-indole
(3S,4R)-1-(5-fluoro-1H-indole-2-carbonyl)-4-(hydroxymethyl)piperidin-3-ol
(1S,6R)-3-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
4-(5-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl)-2-methylpyridine