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1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(2-phenoxyethyl)piperazine
1-[(2-methoxyphenyl)methyl]-4-[4-(thiophen-3-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
3,5-dimethyl-4-{1-[(2-phenyl-1,3-oxazol-4-yl)methyl]pyrrolidin-2-yl}-1,2-oxazole
3-{2-[(3,4-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}propanoic acid
1-(1H-imidazol-4-ylmethyl)-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
5-{[5-(3,5-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-3-(propan-2-yl)-1,2-oxazole
(4aR,7aS)-1-(2-hydroxyethyl)-4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{[(2-methyl-1H-imidazol-4-yl)methyl](thiophen-2-ylmethyl)amino}ethan-1-ol
(3S,9aR)-3-methyl-8-(quinolin-8-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-methyl-N-[(6-methylpyridin-2-yl)methyl]-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3S,5R)-N5-(2,3-dihydro-1H-inden-5-yl)-N3,N3-dimethyl-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
5-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-4-methyl-2-(propan-2-yl)pyrimidine
(2R,6R)-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
5-benzyl-2-methyl-4-{1-[(E)-2-phenylethenesulfonyl]piperidin-4-yl}pyrimidine
1-(cyclohexylmethyl)-N-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]piperidin-3-amine
4-methyl-2-{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
1-({[(5-ethylpyridin-2-yl)methyl](methyl)carbamoyl}methyl)piperidine-4-carboxamide
1-[2-methoxy-5-({[3-(morpholin-4-yl)propyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
(1R,3S,5S)-3-(4-methoxyphenyl)-8-(1-methyl-1H-pyrrole-2-carbonyl)-8-azabicyclo[3.2.1]octane
N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-1H,4H,6H,7H-pyrano[4,3-c]pyrazole-3-carboxamide
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(methylsulfanyl)ethyl]amine
(1R,5R)-6-benzyl-3-(5-fluoro-2-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane
N,8-dimethyl-N-(2-phenylethyl)-3-(piperidin-1-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
(4aR,7aS)-1-{[3-(hydroxymethyl)-2,4,6-trimethylphenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(2,5-dioxoimidazolidin-4-yl)-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}propanamide
2-ethyl-9-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 3-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]benzoate
N,N-dimethyl-4-[4-(piperidin-3-yl)benzoyl]piperazine-1-carboxamide
2-ethyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]pyrimidine-5-carboxamide
4-({4-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]furan-2-yl}methyl)morpholine
8-(4-chloro-2,6-dimethoxyphenyl)quinolin-4-amine
N-[1-(3-methoxyphenyl)propan-2-yl]-1-(4-methylbenzoyl)piperidin-4-amine
2-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]benzonitrile
4-ethyl-5-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,3-thiazol-2-amine
1-(cyclohexylmethyl)-3-hydroxy-3-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}piperidin-2-one
N-methyl-3-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
methyl 7-oxo-9-[2-(piperidin-1-yl)ethoxy]-3-(thiophene-3-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-({[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[3-(2-fluorophenyl)propyl]-4-(2-oxopyrrolidin-1-yl)butanamide
N-benzyl-N-methyl-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-amine
N-{1-[1-(1-methoxypropan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
3-hydroxy-3-{[methyl(pyridin-2-ylmethyl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
5-methyl-4-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)pyrimidine
1-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-4-(1H-imidazol-2-yl)-1H-1,2,3-triazole
1-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-phenylazepane
1-cyclobutanecarbonyl-4-[1-(2-methylphenyl)piperidin-4-yl]-1,4-diazepane
1-methyl-N-[2-(4-sulfamoylphenyl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-1-methylazepane-2-carboxamide
N2-[1-(cyclohex-1-en-1-yl)ethyl]-5-fluoro-N4,N4-dimethylpyrimidine-2,4-diamine
2-[(4-fluorophenyl)methyl]-4-(1H-imidazole-4-carbonyl)morpholine