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1-[2-(piperidin-2-yl)ethyl]-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-1,2,3-triazole-4-carboxamide
3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}-N-[(3S)-2-oxoazepan-3-yl]benzamide
N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-(1-tert-butyl-5-methyl-1H-1,2,4-triazol-3-yl)benzamide
2-(1-cyclopentanecarbonylpiperidine-4-carbonyl)-2,3-dihydro-1H-isoindole
N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)-4-methyl-N-(pyridin-4-ylmethyl)benzamide
N-[(3R,4S)-1-(cyclobutylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetamide
(3S,4S)-4-cyclopropyl-1-[2-(2-oxoazepan-1-yl)acetyl]pyrrolidine-3-carboxylic acid
N-{2-[methyl(phenyl)amino]ethyl}-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-({methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)pyridine-3-carboxylic acid
4-[3-(furan-2-yl)phenyl]-1-[(5-methyl-1H-pyrazol-3-yl)methyl]-1H-1,2,3-triazole
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(5-ethyl-2,6-dimethylpyrimidin-4-yl)pyrrolidin-3-yl]methanol
N-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)-3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
N-{4-[(2-methoxyethyl)carbamoyl]phenyl}-2-methyl-2,7-diazaspiro[4.5]decane-7-carboxamide
4-{[(3-fluorophenyl)methyl]amino}-5-methyl-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
2-(1H-1,2,3-triazol-1-yl)-N-{1,4,6-trimethyl-1H-pyrazolo[3,4-b]pyridin-3-yl}acetamide
2-({4-phenyl-5-[1-(1H-pyrazol-1-yl)ethyl]-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
2-[1-({3-[3-(azepan-1-yl)-2-hydroxypropoxy]phenyl}methyl)piperidin-4-yl]acetamide
N-cyclopentyl-2-(morpholine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
2-(2-methoxyphenyl)-N-[2-(methylsulfamoyl)phenyl]pyrrolidine-1-carboxamide
3-(2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N-cyclohexyl-3-[(1-methyl-3-propyl-1H-pyrazol-5-yl)formamido]propanamide
2-methyl-1-{8-[(4-methylpiperazin-1-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}butan-1-one
N3-benzyl-1-(2-methoxyethyl)-N3-methyl-4-oxo-N5-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-5-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[(2S,4R,5R)-5-(4-chlorophenyl)-1-ethyl-2-methyl-4-{[(pyridin-2-ylmethyl)amino]methyl}pyrrolidin-2-yl]methanol
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
N-[1-(6-chloro-2-methylquinoline-4-carbonyl)piperidin-3-yl]acetamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[(4-ethylphenyl)methyl]-N-methylacetamide
3-[(3-hydroxypiperidin-1-yl)methyl]-N-(1-methyl-1H-pyrazol-4-yl)benzamide
N-[1-(1-cyclopentylpiperidin-4-yl)-1H-pyrazol-5-yl]benzamide
3-(2H-1,3-benzodioxol-5-yl)-5-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-3,5-difluoropyridine
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-(3-methylbut-2-en-1-yl)piperazin-2-one
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-4-hydroxy-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-methyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3S,4S)-1-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(piperidin-1-yl)pyrrolidin-3-ol
N-[(4-fluorophenyl)methyl]-3-[1-(1H-imidazole-5-carbonyl)piperidin-4-yl]propanamide
3-[(4-hydroxy-6-methylpyrimidin-2-yl)methyl]-7-methyl-3H,4H-thieno[3,2-d]pyrimidin-4-one
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2,3-dimethylquinoxaline-6-carboxamide
2-(1-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}azetidin-3-yl)pyridine
5-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidine-1-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
(4aR,7aS)-1-acetyl-4-[(4-ethoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(4-{[2-(cyclopentyloxy)phenyl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
2-[4-(2H-1,3-benzodioxol-5-yl)-2-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy]-1-[4-(4-fluorophenyl)piperazin-1-yl]ethan-1-one
2-(2-{1-oxa-7-azaspiro[3.5]nonan-7-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
(1S,5R)-3-(2-cyclopentylacetyl)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}-4-(pyridin-4-yl)piperidine-1-carboxamide
5-[2-(piperidin-1-yl)ethyl]-7-[({[2-(trifluoromethyl)phenyl]methyl}amino)methyl]-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one