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(2R)-2-[(3-methyl-1-propyl-1H-pyrazol-4-yl)formamido]-3-(pyridin-4-yl)propanoic acid
[1-(2,1,3-benzoxadiazol-5-ylmethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
N-cyclohexyl-N-methyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
6-ethyl-N,1-dimethyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[2-(1H-pyrazol-1-yl)ethyl]-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidine
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1H-imidazol-1-yl)ethyl]acetamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-amino-4-methyl-1,3-thiazole-5-carboxamide
2-({[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)ethan-1-ol
7-(1,3-benzothiazol-2-yl)-4-[(2,6-difluorophenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl 5-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-5-oxopentanoate
N-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
(5S,9aS,9bS)-5-(6-methoxy-2H-chromen-3-yl)-2-(2-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-benzyl-3-ethyl-1-{[2-(2-hydroxyethoxy)phenyl]methyl}-1,4-diazepan-5-one
2-[1-(3,6-dimethylpyrazin-2-yl)piperidin-3-yl]-1H-1,3-benzodiazole
N-{[5-(4-chloro-2-fluorophenyl)furan-2-yl]methyl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
2-fluoro-N,4-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]benzamide
7-oxo-N-{[3-(trifluoromethoxy)phenyl]methyl}-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
5-[3-(aminomethyl)pyrrolidin-1-yl]-2-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-2,3-dihydropyridazin-3-one
4-(4-benzylpiperazin-1-yl)-2-methyl-5-propylpyrimidine
1-{1-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea
1-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}piperidine
N-(1-methylpiperidin-4-yl)-4-oxo-4-phenyl-N-(pyridin-4-ylmethyl)butanamide
1-benzyl-3-(2-methoxyethyl)-8-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]acetamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
1-cycloheptyl-4-{[(1,2-dimethyl-1H-imidazol-5-yl)methyl]amino}pyrrolidin-2-one
(2R,3R)-3-[butyl(methyl)amino]-1'-(pyridin-3-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-{8-[(4-acetamidophenyl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
2-[(2S,4S)-2-(diethylcarbamoyl)-4-(dimethyl-1,3-oxazole-5-amido)pyrrolidin-1-yl]acetic acid
3-[5-oxo-3-(3,3,3-trifluoropropyl)-4,5-dihydro-1H-1,2,4-triazol-4-yl]propanoic acid
2-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}acetamide
3-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}phenol
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,3-thiazol-2-yl)piperidine
6-(quinolin-6-yl)pyrazine-2-carboxylic acid
2-(6-fluoro-2-oxo-1,2-dihydroquinoline-4-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-(1-ethyl-1H-imidazol-2-yl)-1-methanesulfonylpiperidine
1-[(4-fluorophenyl)methyl]-N-(furan-2-ylmethyl)-N-(prop-2-yn-1-yl)-1H-1,2,3-triazole-4-carboxamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,4-dimethyl-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
5-benzamido-1-cyclopentyl-N-[3-(propan-2-yloxy)propyl]-1H-1,3-benzodiazole-7-carboxamide
1-{4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
3-(furan-3-ylmethyl)-5-(3-methylbutyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
ethyl 5-[({1-[4-(2-phenoxyacetamido)phenyl]piperidin-4-yl}amino)methyl]furan-2-carboxylate
3-methyl-8-[5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-ethyl-5-{3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-2-one
6-(methylamino)-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
N,N-diethyl-1-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
6-methyl-5-{2-oxo-2-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-({5-[(4-methoxy-2-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea