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1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-2-(1,3-thiazol-2-yl)piperidine
5-methyl-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-N-(2-methoxyethyl)-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][(1-ethylpyrrolidin-2-yl)methyl]{[1-(2-methoxyethyl)piperidin-4-yl]methyl}amine
[(5-{[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]methyl}thiophen-3-yl)methyl]dimethylamine
1-(3-ethoxyphenyl)-3-[2-(1-hydroxycyclopentyl)ethyl]-3-methylurea
3-(3-fluorophenyl)-4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-1-(4-methoxyphenyl)-1H-pyrazole
(3R,4R)-4-(azepan-1-yl)-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-3-ol
{3-ethyl-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}methanol
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-2-(pyridin-2-yl)acetamide
2-[5-(5-methyl-4,5,6,7-tetrahydro-2H-indazol-3-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl]acetamide
2-[4-(2-chlorophenyl)-4H-1,2,4-triazol-3-yl]ethan-1-amine
N-ethyl-N'-(3-ethylphenyl)-N-[(5-methylfuran-2-yl)methyl]butanediamide
2-{imidazo[1,2-a]pyridin-3-yl}-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[(1R,3R)-3-aminocyclopentyl]-N'-(3-hydroxyphenyl)butanediamide
N-[3-(4-chlorophenoxy)-2-hydroxypropyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{4-[(2-fluorophenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-3-methylbutanamide
3-{[(3S,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}phenol
2-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}(methyl){[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amine
2-{[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-6-methoxyphenol
6-ethyl-N-(furan-2-ylmethyl)-2-(morpholin-4-yl)pyrimidin-4-amine
2-ethyl-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidine-5-carboxamide
3-(1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}piperidin-3-yl)-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-methyl-8-[(2,4,6-trimethoxyphenyl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(1,3-benzothiazole-2-carbonyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
2-[3-(furan-2-yl)-5-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
5-chloro-6-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]pyridine-3-carboxylic acid
3-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}piperidine-1-carboxamide
5-methyl-4-({2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}methyl)-2-(3-methylthiophen-2-yl)-1,3-oxazole
N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)thian-4-amine
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]ethan-1-one
(4aS,8aR)-6-(2-cyclopropylacetyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-[2-(2-chlorophenyl)ethyl]-2-(methoxymethyl)-N,6-dimethyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidine-1-carbonyl}phenol
2-hydroxy-N,3-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]benzamide
1-(2-methoxy-5-{[4-(methoxymethyl)piperidin-1-yl]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
2-[2-fluoro-3-(pyrrolidin-1-ylmethyl)phenoxy]-5-(trifluoromethyl)pyridine
(2S,4S)-4-amino-1-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}pyrrolidine-2-carboxylic acid
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-4-cyclobutaneamido-N-methylbenzamide
4-[(5-{6-chloroimidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-3-yl)methyl]-1-methylpiperidine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2-(4-hydroxypiperidin-1-yl)acetamide
1-(1-benzothiophene-5-carbonyl)-4-(pyridin-4-ylmethyl)-1,4-diazepane
2-amino-6-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-4-[5-(hydroxymethyl)furan-2-yl]pyridine-3-carbonitrile
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N'-(3,5-dimethylphenyl)propanediamide
4-(3-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane-9-carbonyl}phenyl)-2-methylbutan-2-ol
1,6-dimethyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-[4-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)piperidin-1-yl]-1λ6-thiane-1,1-dione