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2-(dimethyl-1,3-thiazol-5-yl)-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]acetamide
8-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-({1-[(2-cyclohexylpyrimidin-5-yl)methyl]piperidin-4-yl}methyl)acetamide
{1-[(5-chlorothiophen-2-yl)sulfonyl]-4-[(4-methoxyphenyl)methyl]piperidin-4-yl}methanol
4-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholine
[1-(isoquinoline-5-carbonyl)-3-(2-methylpropyl)piperidin-3-yl]methanol
8-[2-(methylsulfanyl)benzoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-phenylpyrrolidin-3-ol
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[2-(1H-pyrazol-1-yl)butanoyl]piperazin-2-one
N-(3-chloro-4-methylphenyl)-3-oxo-3-{9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}propanamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}ethan-1-one
methyl({1-[1-(oxolane-3-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)(propan-2-yl)amine
3-(4-fluoro-3-methylphenyl)-5-(morpholine-4-sulfonyl)benzoic acid
4-{[(1R,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzoic acid
2,7,8-trimethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]quinoline-4-carboxamide
3-ethyl-8-{[4-(3-hydroxyprop-1-yn-1-yl)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-methyl-4-{2-[1-(2-phenylethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}piperazine
(1-{5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-3-yl)methanol
2-[(3,5-difluorophenyl)methyl]-8-(2-hydroxyacetyl)-2,8-diazaspiro[4.5]decan-3-one
3-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide
2-chloro-N-[2-(3,4-dimethoxyphenyl)ethyl]-5-acetamidobenzamide
2-{[1-(oxane-2-carbonyl)piperidin-4-yl]oxy}pyrimidine
N3-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
2-(ethylamino)-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)pyrimidine-5-carboxamide
2-[4-(7-methoxy-3,7-dimethyloctyl)-1-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
{3-[(3-chlorophenyl)methyl]-1-[(2,4,6-trimethoxyphenyl)methyl]piperidin-3-yl}methanol
N-(2-methylphenyl)-N'-[(1R)-1-phenylethyl]propanediamide
9-(1,4-dithiepan-6-yl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-[(1S,2R)-2-phenylcyclopropyl]-4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
5-methanesulfonyl-1'-(1-methyl-1H-pyrrole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-({[3-(1H-pyrazol-1-yl)phenyl]methyl}(pyridin-2-ylmethyl)amino)butan-1-ol
ethyl 1-[(3-hydroxyphenyl)methyl]-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
methyl 3-(cyclohex-3-ene-1-carbonyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-propyl-4-{6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}piperazine
N-({5-[(5-propylfuran-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
3-methyl-1-(2-methylpropyl)-4-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]piperazin-2-one
N-{1-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidin-3-yl}acetamide
2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-4-amine
1-{6-methyl-5-[5-(trimethyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}ethan-1-one
1-{[3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazin-1-yl]methyl}naphthalen-2-ol
5-{[4-(adamantan-1-yl)piperazin-1-yl]methyl}-N-propylpyrimidin-2-amine
N-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methyloxolan-3-amine
3-(1-ethyl-1H-imidazol-2-yl)-1-[3-(3-methoxyphenoxy)propyl]piperidine
5-methanesulfonyl-1'-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-{4-[2-(2-aminopyrimidin-5-yl)-1H-imidazol-1-yl]phenyl}-1H-pyrazole-5-carboxylic acid
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)imidazo[1,2-a]pyridine-3-carboxamide
4,6-dimethyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrimidin-2-amine
4-{2-oxo-8-[2-(1H-pyrazol-1-yl)butanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}butanoic acid
3-(4-chloro-2-methylbenzoyl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine
8-(6-methylpyridazin-3-yl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one