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5-fluoro-N-methyl-N-[3-(oxolan-2-yl)propyl]quinazolin-4-amine
4-[(3-aminopyrrolidin-1-yl)sulfonyl]-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
4-(2-methoxyethyl)-N-[4-(2-methoxyphenyl)phenyl]piperazine-1-carboxamide
3-{1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]piperidin-3-yl}propanoic acid
5-(3-phenylpropyl)-5-(piperidin-4-yl)-3-(pyridin-4-ylmethyl)imidazolidine-2,4-dione
1-[(dimethyl-1,3-thiazol-5-yl)methyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-cyclobutyl-6-(4-fluorophenyl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carboxamide
2-(3-fluorophenyl)-N-[(7-{[5-(methoxymethyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]acetamide
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}-2-methylpiperidine
7-chloro-4-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
(4aR,7aS)-1-(cyclopropylmethyl)-4-(2-methoxy-6-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-1-(3-methoxyphenyl)piperazin-2-one
2-(2,4-difluorobenzoyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-fluoro-N-({1-[3-(methylsulfanyl)propanoyl]piperidin-3-yl}methyl)benzamide
3-chloro-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-6-methyl-N-(propan-2-yl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
(4aR,7aS)-1-propanoyl-4-(pyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopropyl-N-(1-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
6-chloro-N-(1,4-oxazepan-6-ylmethyl)imidazo[2,1-b][1,3]thiazole-5-sulfonamide
2-(cyclopropylmethyl)-N-[(3-fluorophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
(1S,5R)-3-[(5-chloro-2,4-dimethoxyphenyl)methyl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidine-1-sulfonamide
4-amino-5-(2H-1,3-benzodioxol-4-yl)-2-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[2,3-d]pyrimidin-7-one
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]formamido}acetic acid
3-(4-methyl-2-oxo-1,2-dihydroquinolin-3-yl)benzoic acid
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(2-methylpropyl)piperidine-4-carboxamide
4-(2-methoxy-4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}phenoxy)-1-methylpiperidine
1-[(5-methylthiophen-2-yl)methyl]-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(2-fluorophenoxymethyl)piperidine
dimethyl({4-methyl-5-[1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
N,N-dimethyl-1-[3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)benzenesulfonyl]pyrrolidin-3-amine
(1S,5R)-6-(furan-3-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3aS,6aR)-5-(4-amino-5-methylpyrimidin-2-yl)-3-[2-(3-chlorophenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-{1'-[(2-methoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
(1,4-dioxan-2-ylmethyl)(methyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)piperidin-4-amine
4-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-1λ6-thiomorpholine-1,1-dione
1-ethyl-2-oxo-N-[2-(3-phenylpiperidin-1-yl)ethyl]-1,2-dihydropyridine-4-carboxamide
2-[(2,5-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
N-[(2-methoxyphenyl)methyl]-N-propyl-1H-1,2,4-triazole-5-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(furan-2-carbonyl)piperidin-3-yl]piperazine
N-[1-(2-phenylethyl)piperidin-3-yl]quinoxalin-2-amine
(4aS,8aS)-2-{[2-(propylamino)pyrimidin-5-yl]methyl}-decahydroisoquinolin-4a-ol
2-(3-ethoxyphenyl)-2-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]acetic acid
8-[(2S)-3-hydroxy-2-methylpropyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-[(4aR,8aR)-7-cyclopentanecarbonyl-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-phenylethan-1-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-{[5-(hydroxymethyl)furan-2-yl]methyl}piperazin-2-yl}ethan-1-ol
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(3,5-difluorophenyl)methyl]piperidine-3-carboxamide
4-(1,4-dioxane-2-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol