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5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-3-ylmethyl)pyridin-2-amine
N-[(2S,4R,6R)-2-(9H-fluoren-2-yl)-6-(propan-2-yl)oxan-4-yl]acetamide
(2S)-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}pyrrolidine-2-carboxamide
4-methyl-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-(furan-3-carbonyl)-4-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
(3S,4R)-1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-4-methyl-3-(2-methylpropyl)piperidin-4-ol
1'-(2H-1,3-benzodioxole-5-carbonyl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
1-(4-chlorophenyl)-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)cyclobutane-1-carboxamide
2-(2,3-dimethoxy-5-methylphenyl)-2-[4-(pyrazin-2-yl)piperazin-1-yl]acetic acid
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-methyl-1-(4-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperazin-1-yl)butan-1-one
2-(2,5-dioxoimidazolidin-1-yl)-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}acetamide
methyl 1-{3-[4-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)phenoxy]-2-hydroxypropyl}piperidine-4-carboxylate
2-{[(5-ethyl-2-methylpyrimidin-4-yl)amino]methyl}-3,5-dimethylpyridin-4-ol
N-[(1-methylpyrrolidin-3-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-(pyridin-2-ylmethyl)piperazin-2-yl}ethan-1-ol
4-hydroxy-N-(4-methyl-3-propanamidophenyl)-4-phenylpiperidine-1-carboxamide
N-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)adamantan-1-amine
methyl[(5-methylfuran-2-yl)methyl]{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
3-(1-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
1-(azocan-1-yl)-3-[2-methoxy-4-({[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
1-(2-{4-[2-(furan-2-yl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-methyl-2-(propan-2-yl)pyrimidine-5-carboxamide
N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-2-(4-{7-methylthieno[3,2-d]pyrimidin-4-yl}-1H-pyrazol-1-yl)acetamide
2-({4-methyl-1-[5-(methylcarbamoyl)furan-2-yl]-1H-1,3-benzodiazol-2-yl}methoxy)acetic acid
1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
[(3R,5R)-5-(morpholin-4-ylmethyl)-1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)piperidin-3-yl]methanol
7-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
2-(azepan-1-ylmethyl)-4-(1,3-benzothiazol-2-yl)phenol
{[2-(difluoromethoxy)phenyl]methyl}(methyl)[(2-methylpyridin-4-yl)methyl]amine
1-[2-(3-chloro-4-hydroxyphenyl)acetyl]-2-methyl-1,4-diazepan-5-one
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2-hydroxy-3-(2-methylphenoxy)propanamide
(4aR,8aR)-2-methanesulfonyl-7-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-decahydro-2,7-naphthyridin-4a-ol
[1-(2-chlorophenyl)-2-(2-cyclopropyl-1H-imidazol-1-yl)ethyl]dimethylamine
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-3-(pyrazin-2-yl)propanamide
2-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]-N,6-dimethylpyrimidin-4-amine
4-{3-[3-(1H-imidazol-1-yl)propoxy]phenyl}-1,3-dimethyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-benzyl-N-(4-hydroxybutyl)-2-(2,3,6-trimethylphenoxy)acetamide
2-methoxyethyl 4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carboxylate
N-(1-benzyl-1H-pyrazol-3-yl)-2-[3-(5-methylfuran-2-yl)-1H-pyrazol-1-yl]acetamide
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-methyl-N-(2-phenylethyl)pyridin-2-amine
N-[2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]pyridine-3-carboxamide
(2R,3R)-1'-(furan-3-carbonyl)-3-(1,2,3,6-tetrahydropyridin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-[2-amino-5-(2-carboxyethyl)-6-methylpyrimidin-4-yl]piperidine-3-carboxylic acid
2-[1-(1-cyclobutanecarbonylpiperidine-4-carbonyl)azetidin-3-yl]pyridine
2-[1-(difluoromethyl)-3-methyl-1H-pyrazol-4-yl]benzamide
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amine
(2S,4S)-4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxylic acid