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4-(4-ethyl-1H-pyrazol-5-yl)-1-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]piperidine
N-[5-carbamoyl-2-(2-methylpiperidin-1-yl)phenyl]-4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
3-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)-4,6-dimethyl-1,2-dihydropyridin-2-one
2-(4-{[4-(benzyloxy)phenyl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
(1R,7S)-3-(2,2-dimethylpropyl)-6-(3-oxo-1,4-diazepane-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
(4aS,7aR)-1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(dimethylamino)-2-(3-methylphenyl)-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-6-chloro-N-methylimidazo[1,2-a]pyridine-2-carboxamide
4-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-6-(morpholin-4-yl)pyrimidin-2-amine
N-[4-({3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}methyl)phenyl]acetamide
1,9-dimethyl-4-[2-(propan-2-yl)oxane-4-carbonyl]-1,4,9-triazaspiro[5.5]undecane
1-[7-(3-chlorophenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(3,5-dimethyl-1H-pyrazol-1-yl)propan-1-one
N-[(4-fluorophenyl)methyl]-3-[1-(3-phenylprop-2-ynoyl)piperidin-4-yl]propanamide
methyl[2-(1H-pyrazol-4-yl)ethyl]({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
N-[(1R,3R)-3-aminocyclopentyl]-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
N-(1-{1-[1-(4-chlorophenyl)cyclopropanecarbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
methyl (2S,4S,5R)-4-(benzylcarbamoyl)-5-(2,3-difluorophenyl)-1-methylpyrrolidine-2-carboxylate
1-[(4-methoxyphenyl)methyl]-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-(3-methyl-3-phenylpiperidine-1-carbonyl)-2-(4H-1,2,4-triazol-4-yl)pyridine
2-(1H-imidazol-4-yl)-N-[2-(3-phenylpropoxy)phenyl]acetamide
1-ethyl-2,5-dimethyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1H-pyrrole-3-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]propanamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,2,2,6,6-pentamethylpiperidin-4-amine
3-(1,4-diazepane-1-carbonyl)-N-[(5-methyl-1H-imidazol-4-yl)methyl]benzene-1-sulfonamide
4-(4-chlorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]butan-1-one
2-({[(3R,4R)-4-(hydroxymethyl)-1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[1-(benzenesulfonyl)piperidin-4-yl]-2-(2,3-dihydro-1H-inden-1-yl)acetamide
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]cycloheptanamine
4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]pyrimidin-2-amine
(1R,5R)-6-{[4-(propan-2-yl)phenyl]methyl}-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-[3-(1H-indol-3-yl)propanoyl]-1-methylpiperazine-2-carboxylic acid
N-[3-(cyclohexylcarbamoyl)-2-methylphenyl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}-2-(1-methyl-1H-imidazol-2-yl)piperidine
1-(3-{2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}propyl)pyrrolidin-2-one
1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2-(pyridin-4-ylsulfanyl)ethan-1-one
2-cyclopentyl-1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
4-(1-ethyl-1H-pyrazol-4-yl)-1-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1H-1,2,3-triazole
4,4,4-trifluoro-1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]butan-1-one
3-[3-({cyclopropyl[(2-methoxyphenyl)methyl]amino}methyl)-1H-indol-1-yl]propanamide
[2-ethoxy-5-(1H-imidazol-2-yl)phenyl]methyl acetate
(2S,4S)-4-{[(2-chlorophenyl)methyl]amino}-1-[(2,3-dimethoxyphenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
1-(4-methyl-1,2,5-oxadiazol-3-yl)-4-[3-(2-phenylethyl)-1,2-oxazole-5-carbonyl]piperazine
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-1-methyl-1H-pyrrole-2-carboxamide
2-{[2-(trifluoromethyl)morpholin-4-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
3-(carbamoylamino)-N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}propanamide
4-[5-(1H-imidazol-4-ylmethyl)-3-(oxan-4-yl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]pyridine
4-chloro-N-[(3R,4R)-3-hydroxypiperidin-4-yl]-3-methylbenzamide