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N2,N2-dimethyl-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidine-2,4-diamine
3-{ethyl[(1-methyl-1H-imidazol-2-yl)methyl]sulfamoyl}-N-(2-fluoroethyl)benzamide
N-cyclopropyl-N-{2-phenyl-1-[1-(thiophen-3-ylmethyl)piperidin-4-yl]ethyl}pyridine-2-carboxamide
1-{5-[(6-chloropyridin-2-yl)amino]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-2-yl}piperidin-4-ol
2-{N-methyl-2-[1-(propan-2-yl)piperidin-4-yl]acetamido}-2-(thiophen-2-yl)acetic acid
2-(1H-indol-4-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(3S,4R)-4-(2-methoxyphenyl)-1-[3-(morpholin-4-yl)propanoyl]pyrrolidine-3-carboxylic acid
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-ol
5-{1-[1-(3-methylpyridin-2-yl)propan-2-yl]-1H-1,2,3-triazol-4-yl}pyrimidine
N-{[7-(5-acetylthiophen-2-yl)-1H,2H-naphtho[2,1-b]furan-2-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
1-[(2-chlorophenyl)methyl]-N-[2-methyl-2-(morpholin-4-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
5-{2-[2-(propylsulfanyl)pyrimidin-5-yl]-1H-imidazol-1-yl}-1H-1,2,3-benzotriazole
2-{2-[(1R,5S)-6-azabicyclo[3.2.1]octan-6-yl]-2-oxoethyl}-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
5-acetyl-N-[(3-methyloxetan-3-yl)methyl]thiophene-2-carboxamide
4-{4-[2-(2-methoxyphenyl)pyrrolidin-1-yl]piperidin-1-yl}-N-[2-(morpholin-4-yl)ethyl]benzamide
(1S,5R)-6-(3-chlorothiophene-2-carbonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-(3-hydroxy-3-methylbutyl)-N-[(6-hydroxypyrimidin-4-yl)methyl]benzamide
N-[2-(dimethylamino)ethyl]-4,6-dimethyl-2-oxo-N-(oxolan-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
N-(2,3-dimethylphenyl)-N'-[3-(morpholin-4-yl)propyl]propanediamide
6-cyclopentyl-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]-2-(4-methylphenyl)pyrimidin-4-ol
2-(3-{[methyl(1H-pyrazol-5-ylmethyl)amino]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
1-[6-hydroxy-4-(4-methyl-1H-imidazole-2-carbonyl)-1,4-diazepan-1-yl]ethan-1-one
(2S)-2-({2-[(4-benzylpiperazin-1-yl)methyl]-1,3-oxazol-4-yl}formamido)-3-methylbutanamide
4-(2,4-dioxoimidazolidin-1-yl)-N-[(1-hydroxycyclohexyl)methyl]benzamide
N-{2-[1-(2,3-dimethylphenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
1-[2-(2,5-dimethylphenyl)acetyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
methyl 3-benzamido-5-(benzylamino)-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-1H-1,2,3-triazole-5-carboxamide
(8R,9aS)-8-hydroxy-2-(1H-indol-4-ylmethyl)-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
1-[1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carbonyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
2-[3-(2-hydroxyethyl)-4-(2-phenylethyl)piperazin-1-yl]-6-methylpyridine-3-carboxamide
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1H-1,2,3-benzotriazole-5-carboxamide
ethyl 3-[(3-chlorophenyl)methyl]-1-(6-methylpyridine-3-carbonyl)piperidine-3-carboxylate
ethyl 5-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-[2-(dimethylamino)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
N-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]-4-methylbenzamide
1-[(2,3-dichlorophenyl)methyl]piperidine-3-carbonitrile
1-[(4-chloro-2-fluorophenyl)methyl]azepan-4-amine
1-[2-methyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-{1-oxaspiro[4.4]nonan-3-yl}urea
3-ethyl-5-{[5-(1-ethyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-4,5-dihydro-1,2-oxazole
N-butyl-N-(3-phenylprop-2-yn-1-yl)quinoxaline-5-carboxamide
5-benzyl-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[(1,4-dimethylpiperazin-2-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[2-(furan-2-yl)ethyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]cyclohex-1-ene-1-carboxamide
2-phenyl-7-(pyridine-4-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-cyclopropyl-6-phenyl-N-propylimidazo[2,1-b][1,3]thiazole-3-carboxamide