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1-[(4-hydroxyazepan-4-yl)methyl]-3-phenylurea
1-{2-[(7-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)amino]-4-methylpyrimidin-5-yl}ethan-1-one
3,3-dimethyl-1-[(3S,4R)-1-[2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]urea
[(2S,4R,5R)-4-({[2,2-dimethyl-3-(morpholin-4-yl)propyl]amino}methyl)-5-(2-fluorophenyl)-1-methylpyrrolidin-2-yl]methanol
2-(4-fluorophenoxymethyl)-5-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-carbonyl)pyrimidin-4-ol
2-(2-{[(2,5-dimethylphenyl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)-2-methylpropanoic acid
[(2,2-dimethyloxan-4-yl)methyl](ethyl){[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-methyl-5-[3-(oxan-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-1H-1,3-benzodiazole
N-(2-{1-[6-(dimethylamino)pyrimidin-4-yl]piperidin-4-yl}ethyl)acetamide
5-tert-butyl-N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-1,3,4-oxadiazol-2-amine
8-fluoro-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}quinoline-2-carboxamide
N4-[(2,4-difluorophenyl)methyl]-5-methylpyrimidine-2,4-diamine
4-(4-benzyl-1H-1,2,3-triazol-1-yl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
4-(2,4-dioxoimidazolidin-1-yl)-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}benzamide
3-methyl-N-[1-(pyrimidin-4-yl)ethyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
4-oxo-N-[(1r,4r)-4-hydroxycyclohexyl]-3,4-dihydroquinazoline-2-carboxamide
1-methyl-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl (2S,4S)-4-(2,3-dimethyl-1H-indole-7-amido)-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxylate
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-1-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
8-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
N,5-dimethyl-4-[(prop-2-en-1-yl)amino]-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
3-methyl-7-(3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}propanoyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
methyl 2-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}-1,3-oxazole-4-carboxylate
3-(1H-indazol-1-yl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
2-(3-methoxyphenyl)-N-[1-(pyridin-4-yl)propyl]-1,3-benzoxazole-6-carboxamide
2-{4-[(4-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}-1,3-thiazole-4-carboxamide
2-cyclobutyl-1-[(3R,4R)-4-cyclopropyl-4-hydroxy-3-methylpiperidin-1-yl]ethan-1-one
4-{[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole-3-carboxylic acid
2-(2-chlorophenyl)-3-methyl-N-[(3-methyloxetan-3-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-({3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1H-pyrazole-3-carboxylic acid
N-{[1-(1-benzothiophen-2-ylmethyl)piperidin-3-yl]methyl}-1-phenylmethanesulfonamide
N-ethyl-3-fluoro-4-methoxy-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)benzamide
7-[(4-fluorophenyl)methyl]-2-[(2-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(2-oxoimidazolidin-1-yl)ethyl]benzamide
4-methyl-2-{2-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
2,5-dimethyl-3-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrazine
2-[2-(1H-imidazol-1-yl)ethyl]-1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine
2-(6-chloro-2H-1,3-benzodioxol-5-yl)-8-methoxy-5-[(4-methyl-1H-imidazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
3-[(2-fluorophenyl)formamido]-N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}propanamide
N-(4-{[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(4-fluorophenyl)ethyl)piperidin-1-yl]methyl}phenyl)acetamide
1-(1-methyl-1H-indole-2-carbonyl)-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
3-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-2-(4-methoxyphenyl)-7-methylquinoline
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}benzamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2,3,4-trimethoxybenzamide
7-[(4-chlorophenyl)methanesulfonyl]-2-oxa-7-azaspiro[4.5]decane
1-[3-(2-chlorophenoxy)azetidin-1-yl]-3-(pyridin-2-yl)propan-1-one
ethyl 4-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate
4-benzyl-1-(1,3-dihydroxypropan-2-yl)-3-ethyl-1,4-diazepan-5-one
(1S,6R)-9-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-3,9-diazabicyclo[4.2.1]nonane
3-[2-(2-methoxyethyl)morpholin-4-yl]-N-(2-methylphenyl)-3-oxopropanamide