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(3S)-3-fluoro-1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]pyrrolidine
3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}-N-(2-chlorophenyl)propanamide
(1S,5R)-3-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonane
8-(2-{[(2-methylphenyl)methyl]sulfanyl}acetyl)-2,8-diazaspiro[4.5]decan-3-one
N-{[4-(cycloheptyloxy)-3-methoxyphenyl]methyl}-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
1'-(2-hydroxyethyl)-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-5-(methoxymethyl)furan-2-carboxamide
N-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-chlorobenzamide
2-(3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)-6-methylpyridine
1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-phenylbutan-1-one
4-(6-methoxypyrimidin-4-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[4-(3-methylphenyl)phenyl]-1-[(2E)-3-(pyridin-4-yl)prop-2-enoyl]piperidine-4-carboxamide
1-cyclopentyl-N3-methyl-N5-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-[(2-fluorophenyl)methyl]-1-[2-(methylsulfanyl)benzoyl]-1,4-diazepan-5-one
1-methyl-4-phenyl-3-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amino]ethan-1-ol
8-(5-ethoxyfuran-2-carbonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[(2-hydroxyadamantan-2-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N,2-dimethyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-(2,4-dimethoxybenzoyl)-7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{5-[1-(4-fluorobenzenesulfonyl)pyrrolidin-2-yl]-3-methyl-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-methyl-N-[2-(oxan-2-yl)ethyl]-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
N-[2-(2,5-dimethylphenoxy)ethyl]-N-methyl-2-(morpholin-3-yl)acetamide
5-ethyl-2,3-dimethyl-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-[(3R,4R)-4-[2-(2,4-dimethoxy-3-methylphenyl)-1H-imidazol-1-yl]oxolan-3-yl]piperidine
4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine
2-{2-methyl-7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carbonyl}-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
(2S,4S)-N-ethyl-4-(3-hydroxybenzamido)-1-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
(1S,5R)-6-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-(4-{[4-(1-ethylpiperidine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
N-[2-(4-hydroxyphenyl)ethyl]-2-(1-methylpiperidin-2-yl)acetamide
2-[1-(4-phenoxybutanoyl)pyrrolidin-3-yl]benzoic acid
5-(5-chloro-2-methoxypyridin-4-yl)furan-2-carboxamide
2-{[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}benzoic acid
3-{3-[5-(1-ethyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyridine
3-[(6-amino-2-{[(4-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)amino]-1-(pyrrolidin-1-yl)propan-1-one
(3S,4R)-3-benzyl-4-methyl-1-(3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-ol
(2S,4R)-1-(1-ethylpiperidin-4-yl)-4-(furan-3-amido)-N-methylpyrrolidine-2-carboxamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-4-(2-methoxyphenyl)-6-methyl-1,2,3,4-tetrahydropyrimidin-2-one
ethyl 2-({5-oxo-1,4,9-triazaspiro[5.5]undecane-9-carbonyl}amino)benzoate
(1S,5R)-6-(2,5-dimethylfuran-3-carbonyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
(2S,4S)-4-amino-N,N-diethyl-1-[2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetyl]pyrrolidine-2-carboxamide
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
5-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-hexyl-8-[2-(methylamino)pyridine-4-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]benzene-1,2-diol
5-cyclopropyl-N-[2-(dimethylamino)ethyl]-3-methyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-4-carboxamide
1-(7-fluoro-2-methylquinoline-4-carbonyl)pyrrolidin-3-ol
8-chloro-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}quinoline-2-carboxamide
1-{1-[(3-ethoxyphenyl)methyl]piperidin-3-yl}-4-(4-methoxyphenyl)piperazine