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1-{5-[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]thiophen-2-yl}ethan-1-one
N-[2-(5-methyl-4-{[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamido]methyl}-1,3-oxazol-2-yl)phenyl]benzamide
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-{[(3-fluorophenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
5-(morpholin-4-ylmethyl)-N-[1-(pyrazin-2-yl)propan-2-yl]furan-3-carboxamide
N-(3-hydroxypropyl)-1-(methoxymethyl)-N-(naphthalen-1-ylmethyl)cyclobutane-1-carboxamide
2-amino-1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methylpropan-1-one
ethyl 5-(2-fluoro-5-methoxyphenyl)pyridine-3-carboxylate
2-fluoro-N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]benzamide
3-methyl-3-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1-(2,3,4-trifluorophenyl)urea
N-[3-(hydroxymethyl)-2-methylphenyl]-2-{4-[2-(methylsulfanyl)acetyl]morpholin-3-yl}acetamide
2-[3-(2-methoxyethyl)-5-[(propan-2-ylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
(3E)-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pent-3-en-1-one
5-{[2-(cyclopentyloxy)phenyl]methyl}-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(3,3,5,5-tetramethylcyclohexyl)-3,4-dihydropteridin-4-one
diethyl({[3-(piperazine-1-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl})amine
1-[1-(2-chlorobenzoyl)piperidin-3-yl]-4-(2-fluorophenyl)piperazine
N-({1-[(5-ethylpyridin-2-yl)methyl]piperidin-4-yl}methyl)propane-2-sulfonamide
N-{3-[(4-chlorophenyl)sulfanyl]propyl}-1-ethyl-5-oxopyrrolidine-3-carboxamide
(3S,4S)-1-(benzenesulfonyl)-4-{ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}pyrrolidin-3-ol
5-(methoxymethyl)-N-[2-(pyrrolidin-1-yl)ethyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-(dimethylamino)-2-(4-methylphenyl)-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
3-[2-(dimethylamino)-2-(furan-2-yl)ethyl]-1-(2-fluoro-5-methanesulfonamidophenyl)urea
N-[2-(pyridin-3-yloxy)propyl]-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
[(5-ethylpyridin-2-yl)methyl](methyl){[1-(morpholin-4-yl)cyclohexyl]methyl}amine
(3R,4R)-1-{[3-(methylsulfanyl)phenyl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-methyl-1,3-benzothiazole-5-carboxamide
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[2-(piperidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
2-(2,4-difluorophenoxy)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
N-{[3-(3-fluorophenyl)oxolan-3-yl]methyl}-4-methyl-1-propyl-1H-pyrazol-5-amine
1-(4-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-1-yl)-2-phenoxyethan-1-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
N-methyl-N-[4-(morpholin-4-yl)butyl]pyrimidin-4-amine
methyl 6-[(3,4-dimethylphenyl)methyl]-2-[(1-methoxypropan-2-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-{[1-(3-methylbut-2-enoyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{2-[4-(1-tert-butyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethyl}azepane
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-(pyridine-4-carbonyl)piperidine-4-carboxamide
(2-{[4-(quinolin-4-ylmethyl)piperazin-1-yl]methyl}phenyl)methanol
3-{1-[3-(4-ethylphenyl)-1H-pyrazole-5-carbonyl]azetidin-3-yl}pyridine
4-(8-chloroquinolin-2-yl)-1-(3,5-dimethylphenyl)piperazin-2-one
N-[(4-fluorophenyl)methyl]-1-methyl-5-[methyl(1,2-oxazol-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(5-{[4-(isoquinolin-1-yl)piperazin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
N,5-dimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-4-phenylbutan-1-one
2-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-[2-(3-chlorophenyl)ethyl]-2-{2-[(dimethylamino)methyl]-4-(pyrimidin-2-yl)phenoxy}acetamide
6-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]-1-methyl-1H-indole
methyl 3-acetamido-1-[2-(4-methoxyphenyl)ethyl]-5-{[(2-methoxyphenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]phenol
4-[(1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-4-yl)methyl]morpholine
2-(2-methoxyethyl)-9-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one