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(3aR,6aR)-2-(3-chloro-4-methylbenzoyl)-5-(2-hydroxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
N-{[1-(2-methoxyacetyl)piperidin-3-yl]methyl}-2-(4-methoxyphenyl)acetamide
2-(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[4-(pyridin-4-yl)piperidin-1-yl]ethan-1-one
(2S,4R)-4-amino-N-(propan-2-yl)-1-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]pyrrolidine-2-carboxamide
1-(2-chlorophenyl)-3-{1-[1-(1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-cyclopropyl-5-[(3S,4R)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-2-(1H-imidazol-1-yl)-N-(oxolan-2-ylmethyl)acetamide
(4aR,7aS)-1-(pyrimidin-2-yl)-4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(4-fluorophenyl)-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-1,2,3,6-tetrahydropyridine
3-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-1,3-diazinane-2,4-dione
(5-{1-[2-(morpholin-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}furan-2-yl)methanol
4-(4-methoxyphenyl)-N-(2-methyl-1H-1,3-benzodiazol-6-yl)piperazine-1-carboxamide
(2S,4R)-N,N-diethyl-4-[2-(4-hydroxyphenyl)acetamido]-1-propylpyrrolidine-2-carboxamide
2-(6-hydroxy-2-methylpyrimidin-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-ethoxy-4-{[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]methyl}phenol
5-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
3-[(4-cyclopentylpiperazin-1-yl)methyl]-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
2-[2-(4-phenyl-1H-imidazol-5-yl)-1H-pyrrol-1-yl]-1,3-thiazole
2-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}benzonitrile
5-({methyl[(3-{2-[4-(3-methylthiophene-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amino}methyl)pyrrolidin-2-one
[2-(adamantan-1-yl)ethyl](methyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
(2S)-1-{[2-(3-chlorophenyl)-8-methylquinolin-3-yl]methyl}pyrrolidine-2-carboxamide
5-methoxy-2-{4-[3-(morpholin-4-yl)-3-oxopropyl]piperidine-1-carbonyl}-1,4-dihydropyridin-4-one
5-{5-methyl-12-oxo-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-14-yl}thiophene-2-carboxylic acid
3-(pyridin-3-yl)-N-(2,4,6-trimethylpyridin-3-yl)azetidine-1-carboxamide
N-(pyrimidin-4-ylmethyl)-3-(thiomorpholine-4-carbonyl)benzene-1-sulfonamide
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-2-methyl-4-phenylpiperazine
(2R)-2-amino-3-methoxy-1-[4-(2-methoxyphenoxy)piperidin-1-yl]propan-1-one
(2S)-2-[2-(4-methoxy-2,3-dimethylphenyl)-1H-imidazol-1-yl]-3-methylbutan-1-ol
6-[(4-methylphenyl)methyl]-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
(4aS,8aR)-6-[(6-ethoxypyridin-3-yl)methyl]-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-imidazole-4-carboxamide
1-(4-chlorophenyl)-N-{[1-(3-phenoxypropanoyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)pyrrolidin-3-yl]methanol
N-[2-methyl-1-(7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]furan-3-carboxamide
(1R,5R)-3-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
3-methyl-1-(oxan-2-ylmethyl)-1,2-dihydroquinoxalin-2-one
6-[(2-hydroxy-2-methylpropyl)amino]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-{1-[1-(5-fluoropyridine-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
2-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-acetyl-N-[3-(5-chloro-1H-1,3-benzodiazol-2-yl)propyl]piperidine-3-carboxamide
2-(dimethylamino)-N-(2-methoxyethyl)-N,4-dimethylpyrimidine-5-carboxamide
3-{2-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
4-(4-methyl-1H-pyrazol-1-yl)-1-(6-methylpyridazin-3-yl)piperidine-4-carboxylic acid
1-[(1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)methyl]pyrrolidin-2-one
N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-(pyridin-2-ylmethyl)piperidin-3-amine
9-ethyl-1-methyl-4-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
2-ethyl-5-[4-(2-methoxybenzoyl)piperazine-1-carbonyl]pyrimidine
1-cyclopentyl-4-{[(5-ethyl-2-methylpyrimidin-4-yl)amino]methyl}pyrrolidin-2-one