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N-(3-hydroxy-3-methylbutyl)-N-methyl-2-(pyrrolidin-1-yl)propanamide
(3S,5R)-N3-(4-methylphenyl)-N5-(pyrimidin-4-ylmethyl)piperidine-3,5-dicarboxamide
3-(3-cyanophenyl)-5-(cyclopropylsulfamoyl)benzoic acid
N-(propan-2-yl)-5-(1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}pyrrolidin-2-yl)thiophene-2-carboxamide
N-{4-[4-(1H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-4-amine
5-butyl-1-(3-chlorophenyl)-4-(2-methoxyacetyl)piperazin-2-one
N-(3-chloro-4-fluorophenyl)-3-{1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidin-4-yl}propanamide
5-[(2-chlorophenyl)methyl]-3-(cyclopropylmethyl)-5-[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]imidazolidine-2,4-dione
(1S,6R)-9-(1,6-naphthyridin-5-yl)-3,9-diazabicyclo[4.2.1]nonan-4-one
methyl 2-(1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
methyl 3-{[2-(4-fluorophenoxymethyl)-1,3-oxazol-4-yl]formamido}propanoate
2-methoxy-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1,3,6-trimethyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-(4-fluorophenyl)-N-methyl-4-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}butanamide
1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-3-(pyridin-4-yl)propan-1-one
3-[N-benzyl-1-(3-methoxy-5-methylthiophen-2-yl)formamido]propanamide
N-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-2,3-dihydro-1H-inden-2-amine
5-acetyl-2,4-dimethyl-N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1H-pyrrole-3-carboxamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[4-methyl-3-(5-methylthiophen-2-yl)-1H-pyrazol-1-yl]acetamide
5-{1-[2-(1H-imidazol-1-yl)propyl]-4-phenyl-1H-imidazol-5-yl}-3-methyl-1,2-benzoxazole
1-{5-benzyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}-2,5-dihydro-1H-pyrrole
N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-3-(1H-pyrazol-1-yl)propanamide
3,3-dimethyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)butanamide
N-[(7-{[3-(2-hydroxyethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-5-(methoxymethyl)furan-2-carboxamide
N-[(2,5-dimethoxyphenyl)methyl]-5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
4-(4-chlorophenoxy)-1-(6-methylpyridazin-3-yl)piperidine-4-carboxylic acid
dimethyl({2-[2-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl})amine
4-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}pyrimidin-2-amine
2-methyl-4-[(2E)-3-phenylprop-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-butyl-4-methyl-N-[(2-methylphenyl)methyl]-1H-imidazole-2-carboxamide
1-(2,6-dimethylpyrimidine-4-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-tert-butyl-5-{[4-(2-phenylethyl)-1H-1,2,3-triazol-1-yl]methyl}-1,2,4-oxadiazole
1-(3-hydroxy-4-methylbenzoyl)-3-methylpiperidine-3-carbonitrile
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1-benzothiophene-5-carboxamide
(1s,4s)-4-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]cyclohexan-1-ol
N-[(5-methylpyrazin-2-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
N-[3-(hydroxymethyl)-2-methylphenyl]-4-[(3-methylpiperidin-1-yl)methyl]benzamide
N-[(3S,4R)-1-(2-ethoxyacetyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-[(1-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-1-oxopropan-2-yl)sulfanyl]-6-methyl-3,4-dihydropyrimidin-4-one
1-(3-phenylbutyl)-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
7-[(2,3-difluorophenyl)methyl]-2-methanesulfonyl-2,7-diazaspiro[4.5]decan-6-one
3-{2-oxo-2-[(2S)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]ethyl}-3,4-dihydroquinazolin-4-one
N-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
4-[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]-1-methanesulfonylpiperidine
N-benzyl-5-[4-(6-methylpyridin-2-yl)piperazine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N-{2-[1-(thiophene-3-sulfonyl)piperidin-2-yl]ethyl}acetamide
1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-3,3-diphenylpropan-1-one
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(2-oxopropanoyl)piperidin-3-yl]propanamide
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pyridine-4-carboxamide
1-amino-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)cyclopentane-1-carboxamide