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1'-(1H-indole-5-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5,5-dimethyl-3-{2-oxo-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}imidazolidine-2,4-dione
1-(2-methoxyethyl)-4-(2-phenylpyrrolidine-1-carbonyl)pyrrolidin-2-one
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-3-phenylpyrrolidin-3-ol
7-[(2,3-dimethoxyphenyl)methyl]-2-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2,7-diazaspiro[4.5]decane
N-{2-[1-(quinolin-3-yl)-1H-imidazol-4-yl]ethyl}acetamide
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-3-(pyridin-4-yl)propan-1-one
methyl 1-(2-methoxyethyl)-3-(3-methylbutanamido)-5-[(thian-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{[4-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-N-cyclopropylpyridine-4-carboxamide
3-{[3-(2-methoxyethyl)-1-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl]methyl}-1,3-oxazolidin-2-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-N-methyl-2-[methyl(pyridin-3-ylmethyl)amino]acetamide
1-[9-oxo-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carbonyl]cyclopropane-1-carboxamide
(3S,4S)-1-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]piperidine-3,4-diol
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,2,6-trimethylquinoline-3-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-2-oxo-N-(pyridin-3-ylmethyl)propanamide
3-(1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1H-imidazol-2-yl)-1,2-dihydroquinolin-2-one
5-[1-(2,3-dihydro-1H-inden-2-yl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]-4-methylpyrimidin-2-amine
4-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}methyl)-2,1,3-benzoxadiazole
(2R,3R)-3-{methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-[2-(1H-imidazol-1-yl)acetyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
4-(furan-2-carbonyl)-2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(3-methoxypropyl)-1-methyl-N-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-amine
N-[1-(4-ethoxyphenyl)propyl]-3-(1-methyl-1H-pyrazol-4-yl)propanamide
(3S,4R)-1-{[3-(methylsulfanyl)phenyl]methyl}-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(morpholin-4-yl)ethyl]amine
1-(1-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}ethyl)-4-methylpiperazine
methyl({[3-(2-methylphenyl)phenyl]methyl})({5-[(oxolan-2-ylmethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)amine
dimethyl(3-{4-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-1-yl}propyl)amine
1-{5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-3-amine
6-[3-(3-methylphenoxymethyl)piperidin-1-yl]pyridine-2-carboxylic acid
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
3-benzyl-5-(cyclopent-2-en-1-ylmethyl)-1H-1,2,4-triazole
N-[2-(1,3-benzothiazol-2-yl)ethyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-(3-fluorophenyl)-6,6-dimethyl-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-(furan-2-ylmethyl)-N,1-dimethyl-5-{methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-[2-(1H-imidazol-1-yl)ethyl]-3-(thiomorpholine-4-carbonyl)benzene-1-sulfonamide
1-(4-{3-[2-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[1-(4-fluorophenyl)ethyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
4-{1-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetyl]piperidin-3-yl}benzoic acid
methyl N-{1-[4-(4-methylphenoxy)piperidin-1-yl]-1-oxopropan-2-yl}carbamate
N-[(3,4-difluorophenyl)methyl]-3-[1-(1,3-oxazole-5-carbonyl)piperidin-3-yl]propanamide
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyrrolidine-1-sulfonamide
4-benzyl-3-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperidin-3-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
(3S,7S)-5-[6-(dimethylamino)pyridine-3-carbonyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-(1-cyclopropanecarbonylpiperidin-3-yl)-2-(naphthalen-2-yloxy)acetamide
5-(dimethylamino)-2-{2-oxo-2-[2-(2-phenylethyl)piperidin-1-yl]ethyl}-2,3-dihydropyridazin-3-one