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(3S,4S)-1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
3-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
2-[(1-{2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidin-3-yl)methyl]-1H-1,3-benzodiazole
9-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[3-(1H-imidazol-1-yl)propyl]-9-[2-(methylsulfanyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
(1S,4S)-2-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}-2-azabicyclo[2.2.1]heptane
3-(4-chlorophenyl)-2-[4-(3-methylthiophen-2-yl)-1H-1,2,3-triazol-1-yl]propan-1-ol
1-(2-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}pyrimidin-4-yl)pyrrolidin-3-ol
1-cyclopentyl-N-ethyl-6-oxo-N-(2-phenoxyethyl)piperidine-3-carboxamide
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]morpholine-2-carboxamide
4-(3,5-dimethyl-1H-pyrazol-4-yl)-6-(propan-2-yloxy)pyrimidin-2-amine
(3R,4R)-1-[(6-fluoroquinolin-2-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[2-(trifluoromethyl)phenyl]ethan-1-one
4-[(1S)-1-cyclohexylethyl]-3-cyclopropyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(dimethylamino)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-(3-methylphenyl)acetamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(5-ethylpyridin-2-yl)methyl]pyrrolidin-3-yl]methanol
({1-[1-(3-fluoropyridin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)urea
4-(methoxymethyl)-1-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidine
6-(aminomethyl)-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-methylpyrimidin-4-amine
2-phenyl-N-{1-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
1-(2,2-dimethyloxane-4-carbonyl)-4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-ethyl-N-(oxan-4-yl)-1,3-oxazole-4-carboxamide
N-ethyl-5-(morpholin-4-ylmethyl)-N-(oxan-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-[(3S,4R)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-[3-(3-methylphenoxymethyl)piperidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
1-{2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-4-methyl-1,2,3,6-tetrahydropyridine
1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}-4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazine
2-[(4-ethoxypiperidin-1-yl)sulfonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-benzyl-N-ethyl-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-[5-(2-cyclopropyl-4-methylpyrimidin-5-yl)-3-methyl-1H-1,2,4-triazol-1-yl]acetic acid
N-cyclopropyl-N-({4-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-4-phenylbenzamide
N-{2-[4-({[(8-methoxyquinolin-2-yl)methyl](methyl)amino}methyl)-5-methyl-1,3-oxazol-2-yl]phenyl}thiophene-3-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-[(3-ethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{3-[(3-chlorophenyl)methyl]-5-[(4-ethylpiperazin-1-yl)methyl]-1H-1,2,4-triazol-1-yl}acetic acid
3-(3-methylbut-2-en-1-yl)-1-(pyridin-2-ylmethyl)piperidine-3-carboxylic acid
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidine
N-(3-hydroxy-2,2-dimethylpropyl)-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-(2-methyl-1H-imidazol-1-yl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
4-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-2-one
N-[2-(1H-indol-3-yl)ethyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}acetamide
1-[1-(2-methoxy-6-methylbenzoyl)piperidin-4-yl]pyrrolidin-2-one
N-cyclobutyl-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-(pyridin-3-ylmethyl)-1-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-(furan-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(4-chlorophenyl)methyl]-8-[(1-ethyl-1H-imidazol-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(2-methoxyethyl)({2-[(4-methoxypyrimidin-2-yl)oxy]hex-5-en-1-yl})methylamine