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5-{5-[3-(4-fluorophenyl)propyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
4-(difluoromethoxy)-N-(1,2-oxazol-3-ylmethyl)benzamide
1-[3-(4-phenylbenzoyl)piperidin-1-yl]propan-1-one
1-(4-methoxybutan-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-[2-fluoro-6-(trifluoromethyl)phenyl]-1-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}urea
N-(4-chloro-3-methoxyphenyl)-2-[4-(pyrrolidin-1-yl)piperidin-1-yl]acetamide
2-[2-(butan-2-yl)phenoxy]-N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N-methylacetamide
ethyl 3-[(3-methoxyphenyl)methyl]-1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidine-3-carboxylate
N-[(3S,4R)-1-[3-(1H-indol-3-yl)propanoyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-2-(2-methyl-1H-indol-3-yl)acetamide
(1R,2R,6S,7S)-4-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-4-azatricyclo[5.2.1.02,6]decane
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
1-(cyclopropylmethyl)-5-[2-(methylamino)pyridine-3-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-methoxy-5-[(E)-2-phenylethenyl]pyridine
2-methyl-5-(4-{2-methylthieno[3,2-d]pyrimidin-4-yl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
2-{1-[(4-fluorophenyl)methyl]-4-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-{4-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]piperazin-1-yl}-4,6-dimethylpyridine-3-carbonitrile
2-(3-fluoro-4-phenylphenyl)-1-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]propan-1-one
4-[(dimethylamino)methyl]-1-(2-phenoxybenzoyl)azepan-4-ol
N-methyl-3-({[(2-methylphenyl)methyl](prop-2-en-1-yl)amino}methyl)pyridin-2-amine
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1,2-oxazole-3-carboxamide
3-{[2-(morpholin-4-yl)pyrimidin-5-yl]formamido}-N-(1,3-thiazol-2-yl)propanamide
2-(4-acetylphenoxy)-N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
(2S)-N2-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]pyrrolidine-1,2-dicarboxamide
2-amino-3-ethyl-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-methyl-6-oxo-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
(2S)-2-{[(3-chloro-4-ethoxyphenyl)methyl]amino}propanamide
3-[(oxolan-3-yl)sulfamoyl]-N-[2-(1,3-thiazol-2-yl)ethyl]benzamide
N-(1-{1-[2-(2-methoxyphenoxy)acetyl]piperidin-4-yl}-2-phenylethyl)-N,2-dimethylfuran-3-carboxamide
4-{3-[(2-methylphenyl)methoxy]azetidin-1-yl}pyrimidine
1-(2-phenylpropyl)-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
8-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
4-{5-[(2E)-3-(pyridin-3-yl)prop-2-enoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}benzonitrile
6-chloro-2-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]-N,N-dimethylquinoline-4-carboxamide
2-(5-acetylthiophen-3-yl)-N-[(2-tert-butyl-6-oxo-1,6-dihydropyrimidin-4-yl)methyl]acetamide
N-(3-methyl-1-{7-[(2,4,6-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)acetamide
(4aR,7aS)-1-(2-methylpropanoyl)-4-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4S)-4-[(4-fluorophenyl)sulfanyl]-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1-(quinolin-4-ylmethyl)pyrrolidine-2-carboxamide
1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2-(oxan-2-ylmethoxy)ethan-1-one
3-{2-[1-(2-hydroxybutyl)-1H-1,2,4-triazol-5-yl]ethyl}quinoxalin-2-ol
3-fluoro-N,6-dimethyl-N-[1-(pyridin-3-yl)propyl]imidazo[1,2-a]pyridine-2-carboxamide
2-amino-N-[(1R,3R)-3-aminocyclopentyl]-4-phenylpyrimidine-5-carboxamide
1-(4-acetyl-1,4-diazepan-1-yl)-3-(3-chlorophenyl)-3-(2-hydroxyphenyl)propan-1-one
4-(furan-2-ylmethyl)-3-[1-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
{4-[(4-chlorophenyl)methyl]-1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl}methanol
3-(3-fluoro-4-methoxybenzoyl)-1-(3-methylbut-2-en-1-yl)piperidine
2-(2-phenylethyl)-9-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-(cyclohex-3-en-1-ylmethyl)-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
7-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}quinolin-8-ol
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(propane-2-sulfonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one