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5-{2-[4-(3-chlorophenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-4-(2-methoxyethyl)-1,4-diazepan-5-one
(3R,4R)-1-(3-methylpyrazin-2-yl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
6-[1-(3,5-dimethyl-1H-indole-2-carbonyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
2-{4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}benzonitrile
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
N-(2-methoxyethyl)-7-methyl-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidine-6-carboxamide
N-[2-(6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]-3-phenyl-1,2-oxazole-5-carboxamide
N-[(1S,2R)-2-aminocyclobutyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
(1S,3R)-3-[(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]cyclohexan-1-amine
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-[2-(1H-pyrrol-1-yl)ethyl]piperazine
2-[(4aR,7aS)-6,6-dioxo-4-[2-(pyrazin-2-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
2-hydroxy-1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2-methylpropan-1-one
1-{2-[1-(2-cyclopentylacetyl)piperidin-2-yl]ethyl}-N-cyclopropyl-1H-1,2,3-triazole-4-carboxamide
2-amino-4-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]amino}quinazoline-6-carboxylic acid
2-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-1-(propan-2-yl)pyrrolidine-3-carboxamide
9-(2-ethylpyridine-4-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-({[(3R,4R)-1-(4-chlorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-cyclohexyl-3-cyclopropyl-5-({[2-(pyrrolidin-1-yl)ethyl]sulfanyl}methyl)-1H-1,2,4-triazole
3-chloro-N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-4-fluoro-1-benzothiophene-2-carboxamide
1-(3-methylpyridin-2-yl)-4-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]piperazine
3-({ethyl[2-(4-methylbenzenesulfonyl)ethyl]amino}methyl)pyrrolidin-3-ol
5-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-1-propylpiperidin-2-one
N-ethyl-2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-(2-methylprop-2-en-1-yl)acetamide
5-(4-ethoxy-3-methoxyphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-(2-methoxy-4-methylphenoxymethyl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-7-acetamido-1-[(4-fluorophenyl)methyl]-N-methyl-1H-1,3-benzodiazole-5-carboxamide
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-N-[2-(ethanesulfonyl)ethyl]acetamide
1-(4,6-dimethylpyrimidin-2-yl)-N-[2-(2-methylpropanesulfonyl)ethyl]piperidin-4-amine
1-[7-(1-benzothiophen-3-yl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
2-[1-methyl-4-(pyridin-4-ylmethyl)piperazin-2-yl]ethan-1-ol
4-(6-ethylpyrimidin-4-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(pyrimidin-2-yl)-N-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-3-amine
N-ethyl-5-methoxy-1,2-dimethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-indole-3-carboxamide
7-methoxy-3-{[4-(prop-2-en-1-yl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-[2-(1H-indol-3-yl)ethyl]-2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-[2-(3-methoxyphenyl)-1-[1-(quinoxaline-6-carbonyl)piperidin-4-yl]ethyl]-N-methylfuran-2-carboxamide
2-(furan-2-yl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-oxoacetamide
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-(2-oxopyrrolidin-1-yl)butanamide
(1S,5R)-6-(2-methoxyethyl)-3-{[5-(4-methylphenyl)furan-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
(4aR,7aS)-N,N-dimethyl-4-(oxane-4-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-[(5-chloro-2,3-dimethoxyphenyl)methyl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
5-{[(5-chlorothiophen-2-yl)methyl]amino}-1-ethyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-methyl-10-oxo-9-(prop-2-en-1-yl)-N-(thiophen-2-ylmethyl)-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-1-methyl-5-phenyl-1H-pyrazole-3-carboxamide
{[(3R,4S)-4-cyclopropyl-1-(4,4,4-trifluorobutyl)pyrrolidin-3-yl]sulfamoyl}(ethyl)methylamine
6-oxo-1-[2-(pyridin-2-yl)ethyl]-N-[3-(pyridin-2-yl)propyl]piperidine-3-carboxamide
ethyl 4-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]piperidine-1-carboxylate
6-methyl-2-[1-(3-phenyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole