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1-[(3-methyl-1-benzofuran-2-yl)methyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
1-(2,3-dimethylphenyl)-4-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}piperazine
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-[(1-methyl-1H-imidazol-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-N-cyclohexyl-5-cyclopropyl-1H-pyrazole-4-carboxamide
4-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
N-{[3-(difluoromethoxy)phenyl]methyl}-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-[2-(4-methylphenyl)ethyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-[cyclohexyl(methyl)amino]-3-[2-({ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
2-[5-cyclopropyl-4-(4-ethylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-(2,5-dimethoxyphenyl)pyrimidine
3-methyl-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}thiophene-2-carboxamide
N-[1-(5-{[2-(4-fluorophenoxy)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(2-oxopyrrolidin-1-yl)benzamide
ethyl 2-{1-[4-(1H-pyrazol-1-yl)butanoyl]piperidin-2-yl}acetate
5-cyclopropanecarbonyl-1'-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzamide
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
methyl (2S,4R)-1-methyl-4-(9-oxo-9,10-dihydroacridine-4-amido)pyrrolidine-2-carboxylate
4-{1-[2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]azetidin-3-yl}morpholine
4-(1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidine
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-(2-methylpropyl)pyridin-2-amine
(4aR,7aS)-1-(2-methoxyacetyl)-4-[2-(thiophen-2-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4R)-4-amino-1-[3-(2-oxopiperidin-1-yl)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-amino-4-(6-methylquinolin-5-yl)-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
1-{2-[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]ethyl}pyrrolidin-2-one
(3R,4R)-1-[(3,4-difluorophenyl)methyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
3-{[6-(2-chlorophenyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazin-2-yl]formamido}propanamide
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
[(3S,5R)-1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
2-[2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamido]-N-methylacetamide
2-({3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-6-ethoxyphenol
8-fluoro-N-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]quinoline-2-carboxamide
1-(furan-2-carbonyl)-4-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperazine
1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(4-hydroxyphenyl)propan-1-one
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{[(3-methylthiophen-2-yl)methyl]amino}benzamide
1-(2-cyclopropylpyrimidine-5-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
4-benzyl-3-ethyl-1-(quinoline-3-carbonyl)-1,4-diazepan-5-one
4-[3-(propan-2-yloxy)phenyl]thiophene-2-carboxamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-methylpropanamide
1-cyclopropyl-3-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}-3-(4-phenylphenyl)pyrrolidine-2,5-dione
3-[(3S,7S,8aS)-3-(cyclohexylmethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-ethylphenyl)urea
(3aR,6aR)-2-acetyl-5-(2-{[(4-methylphenyl)methyl]carbamoyl}ethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(ethylamino)-N-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}-N-methylpyrimidine-5-carboxamide
5-[2-(aminomethyl)piperidine-1-carbonyl]-2-(4-methylphenyl)pyrimidin-4-ol
4-(4-chlorophenyl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]butanamide
2-(1H-imidazol-2-yl)-N-[2-(4-methoxyphenyl)ethyl]benzamide
N-[2-(7-{[3-(2-hydroxyethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-4-methoxybenzamide
4-[2-(methylsulfanyl)propyl]-1-[(4-phenyloxan-4-yl)methyl]-1H-1,2,3-triazole
(3aR,6aR)-2-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5,7-dimethyl-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]pyrido[2,3-d]pyrimidin-4-amine
3-{1-[(2,5-difluorophenyl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
1-[1-ethyl-5-(2-methoxybenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine