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N-(2-methoxyethyl)-5-methyl-4-[(prop-2-en-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
7-[2-(3-acetyl-1H-indol-1-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-ethyl-3-(1-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-1,2,3-triazol-4-yl)piperidine
(3S,4R)-1-{2-[benzyl(methyl)carbamoyl]ethyl}-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
N-{1-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxy-2-phenylacetamide
N-methyl-5-phenyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-3-carboxamide
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-4-(4-methylpiperazin-1-yl)pentan-1-one
(3S,4R)-1-[2-(benzenesulfonyl)ethyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
N-({3-methyl-7-[(2E)-2-methylbut-2-enoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-sulfonamide
3-({3-ethyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)benzonitrile
1-[1-(2-methoxyethyl)piperidine-3-carbonyl]-4-[(2-methoxyphenyl)methyl]piperazine
1-methyl-4-[7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]-1,4-diazepane
N-(1-{7-[2-(4-chlorophenoxy)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)pyridine-2-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-1-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl}ethan-1-one
methyl 4-({[1-(4-methylquinazolin-2-yl)piperidin-4-yl]formamido}methyl)benzoate
2-chloro-5-acetamido-N-[2-(1H-indol-3-yl)ethyl]benzamide
(1R,3s,6r,8S)-4-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-azatricyclo[4.3.1.13,8]undecane
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-5-ethyl-1,3-oxazole-4-carboxamide
[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl](methyl)(1H-pyrazol-3-ylmethyl)amine
6-(2-chloro-3-methylbenzoyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-[1-(hydroxymethyl)-9-(1H-imidazol-4-ylmethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
2-acetyl-8-(furan-3-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl 4-({4-[3-(morpholine-4-carbonyl)phenoxy]piperidin-1-yl}methyl)benzoate
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methoxyphenoxy)acetamide
(3R,4S)-4-(5-methylfuran-2-yl)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-3-amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(oxan-4-yl)piperidine-3-carboxamide
2-benzyl-8-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,8-diazaspiro[5.5]undecane
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(trifluoromethyl)phenyl]urea
1-(4-{[methyl({[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}thiophen-2-yl)ethan-1-one
3-(dimethyl-1,2-oxazol-4-yl)-1-{4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}propan-1-one
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
2-(1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-3-yl)benzoic acid
N-(1-{7-[(3-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
5-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1,2-oxazole-4-sulfonamide
(2R,6R)-4-(dimethylsulfamoyl)-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
5-benzoyl-1-(cyclopropylmethyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-ethyl-6-(4-fluorophenyl)-N-(pyridin-4-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
{4-benzyl-1-[1-(2,3-dimethylphenyl)piperidin-4-yl]piperidin-4-yl}methanol
4-{1-[(1-propyl-1H-pyrazol-5-yl)sulfonyl]piperidin-3-yl}benzoic acid
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}acetamide
1-methyl-4-oxo-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}-1,4-dihydroquinoline-3-carboxamide
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
4-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2,3-dihydro-1H-imidazol-2-one
9-ethyl-1-methyl-4-(pyridazin-3-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
5-chloro-3-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-(2-chloro-4-fluorophenoxy)propan-1-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1,2,3-thiadiazole-4-carbonyl)piperidin-3-ol
{9-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3-(furan-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
(4aR,8aS)-6-(1-benzothiophen-2-ylmethyl)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-decahydro-1,6-naphthyridine