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2-[4-({3-[2-hydroxy-3-(piperidin-1-yl)propoxy]-4-methoxyphenyl}methyl)piperazin-1-yl]-N,N-dimethylacetamide
2-methoxy-5-[1-(2-methylpropyl)-4-phenyl-1H-imidazol-5-yl]pyrimidine
ethyl 1-(oxane-4-carbonyl)-3-(3-phenylpropyl)piperidine-3-carboxylate
(8aS)-2-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-ethyl-4-methyl-5-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-1,3-thiazol-2-amine
1-(cyclopropylmethyl)-5-[(3-methylquinoxalin-2-yl)methyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
1-(2-aminoethyl)-N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(3R,4R)-1-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
1-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)-1,4-diazepan-6-ol
N-[(2-ethoxypyridin-3-yl)methyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
3-methyl-1-(2-methylpropyl)-4-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]piperazin-2-one
1-{6-chloro-3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}azepan-3-amine
2-methyl-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,3-thiazole-4-carboxamide
N-benzyl-4-methyl-1,4-diazepane-1-sulfonamide
(2S,4R)-4-[4-(3,5-difluorophenyl)-1H-1,2,3-triazol-1-yl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]benzamide
2-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-6-methylphenol
2-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-1,3-benzothiazole
N-[(5-{[2-(5-methylfuran-2-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
7-(2-hydroxyethyl)-2-[2-(1H-indol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-(3-ethoxy-2-hydroxypropyl)acetamide
2-(3-chlorophenyl)-1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-hydroxyethan-1-one
(2S,4S)-N,1-diethyl-4-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamido]pyrrolidine-2-carboxamide
2-hydroxy-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{1-[(2-ethoxyphenyl)methyl]-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
(1S,6R)-3-[(2-cyclohexylpyrimidin-5-yl)methyl]-3,9-diazabicyclo[4.2.1]nonane
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-[1-(4-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
4-(2-aminopyridine-4-carbonyl)-1-phenylpiperazin-2-one
9-[3-(3,5-dimethylphenyl)propanoyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-6-oxo-N-{2-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]ethyl}-1,6-dihydropyridine-3-carboxamide
2-(2-methylphenyl)-1-[3-(pyridin-3-yl)azetidin-1-yl]ethan-1-one
N-({1-tert-butyl-3-[(4-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)acetamide
2-(2-aminoethyl)-N-(2-methoxyethyl)-N-(2-phenoxyethyl)quinazolin-4-amine
4-(2-fluorophenoxy)-1-(3-methylbut-2-enoyl)piperidine-4-carboxylic acid
(4aR,7aS)-4-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
{4-[(5-chlorofuran-2-yl)methyl]-1-methylpiperazin-2-yl}methanol
(1R,7S)-3-[(4-fluorophenyl)methyl]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-methoxy-2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
N-[2-(diethylamino)ethyl]-3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-ethylpropanamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
[(2S,6S)-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-4-phenoxybutanamide
[(3R,4R)-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
3-({2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}(methyl)amino)-1λ6-thiolane-1,1-dione
N-methyl-4-(1H-pyrazol-3-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzamide