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14-(2-hydroxy-8-methylquinolin-3-yl)-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-{[4-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{4-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidine-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
2-methyl-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)pyridine-3-carboxamide
3-[(5-fluoroquinazolin-4-yl)amino]-2,3-dihydro-1λ6-thiophene-1,1-dione
3-(4-methanesulfonylpiperazine-1-carbonyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(pyridin-4-yl)pyridine-3-carboxamide
N-(adamantan-2-ylmethyl)-5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazole-3-carboxamide
methyl 2-(morpholine-4-sulfonyl)-6-(naphthalen-1-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-{[2-(1H-imidazol-4-yl)ethyl]amino}-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[1-(7-{[4-(pyrrolidin-1-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]oxane-4-carboxamide
N-[3-(dimethylamino)propyl]-N,2-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1-(pyridin-2-yl)piperidine-3-carboxamide
N-[(3S)-2-oxoazepan-3-yl]-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)quinoline-2-carboxamide
5-[(diethylcarbamoyl)methyl]-N-ethyl-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(2,5-difluorophenyl)-4-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
4-[2-(2,3-difluorophenyl)acetyl]-1-[(3-methylphenyl)methyl]piperazin-2-one
4-methyl-2-{4-[(2-methyl-1,3-oxazol-4-yl)methyl]piperazin-1-yl}-6-(trifluoromethyl)pyrimidine
3-(1-methylpiperidin-2-yl)-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}propan-1-one
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzamide
4-benzyl-3-ethyl-1-[4-(1H-pyrazol-4-yl)butanoyl]-1,4-diazepan-5-one
8-fluoro-N-[2-(1H-1,2,3-triazol-1-yl)ethyl]quinoline-2-carboxamide
4-[(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
(1R,3S,5S)-8-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
{4-benzyl-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazin-2-yl}methanol
9-methoxy-4-[(4-methoxynaphthalen-1-yl)methyl]-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[2-(2,4-difluorophenyl)ethyl]-1-(ethanesulfonyl)piperidine
7-[4-(4-chlorophenyl)butanoyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)thiomorpholine
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
N-[(2-fluorophenyl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
methyl (2S,4R)-4-(dimethylamino)-1-(2-methoxybenzenesulfonyl)pyrrolidine-2-carboxylate
2-(3-{[8-methoxy-2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenoxy)ethan-1-ol
3-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
6-{1-[3-(dimethylamino)benzoyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
(1R,5S,8S)-N-[2-chloro-5-(morpholin-4-yl)phenyl]-8-hydroxy-3-azabicyclo[3.2.1]octane-3-carboxamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-1-methylpiperidine-4-carboxamide
N-[(2-chlorophenyl)methyl]-3-[1-(furan-2-carbonyl)piperidin-3-yl]propanamide
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]urea
1-ethyl-5-methyl-N-[2-(propan-2-ylsulfanyl)ethyl]-1H-pyrazole-4-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-amine
N-(2-fluorophenyl)-3-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-3-yl}propanamide
N-[(1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)methyl]acetamide
(2S,4R)-4-amino-1-(2,3-dihydro-1-benzofuran-7-carbonyl)-N-ethylpyrrolidine-2-carboxamide
N-[(1S,3R)-3-aminocyclopentyl]-5-cyclopropyl-3-methyl-1H-pyrazole-4-carboxamide
N-{[7-(2,6-dimethylhept-5-en-1-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine-2-carboxamide
(3-benzyl-1H-1,2,4-triazol-5-yl)(3-chlorophenyl)methanol
2-ethyl-4-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}pyrimidine
4-fluoro-3-methyl-N-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}benzene-1-sulfonamide
3-(1-benzofuran-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione