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[1-(3-fluoropyridin-2-yl)-3-propylpiperidin-3-yl]methanol
2,2-dimethyl-5-[4-(pyridin-2-yl)piperazine-1-carbonyl]thiomorpholin-3-one
5-(3-acetylphenoxymethyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
N-(2-fluorophenyl)-3-{1-[2-(morpholin-4-yl)-2-oxoethyl]piperidin-3-yl}propanamide
{5-[1-(1,4-dioxan-2-ylmethyl)-1H-imidazol-2-yl]furan-2-yl}methanol
3-[8-(5-ethylthiophene-3-carbonyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]propanoic acid
8-methoxy-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{[4-(5-amino-3-methyl-1-phenyl-1H-pyrazol-4-yl)phenyl]methyl}acetamide
8-(4-cyclobutyl-6-methylpyrimidin-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{[3-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]methyl}-1,3-benzothiazole
5-{1-[3-(1H-pyrazol-4-yl)benzoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N,N-diethyl-1-{1-[2-(2-methylphenyl)acetyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
2-{1-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-2-yl}pyridine
N-{4-[3-benzyl-3-(hydroxymethyl)piperidine-1-carbonyl]phenyl}acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-propyl-1,3-thiazole-4-carboxamide
N-ethyl-N-[2-(4-methoxyphenoxy)ethyl]-6-methylpyridine-3-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-[2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]piperidin-3-yl]propanoic acid
2,7,8-trimethyl-N,N-bis(prop-2-en-1-yl)quinoline-4-carboxamide
1-{[5,8-dimethoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}piperidine-3-carbonitrile
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
(2S,4R)-4-amino-N,N-diethyl-1-[2-(naphthalen-1-yl)acetyl]pyrrolidine-2-carboxamide
1-[(2,3-difluorophenyl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
2-(2,3-dihydro-1-benzofuran-7-yl)-2-[4-(ethoxycarbonyl)piperazin-1-yl]acetic acid
(2S,4S,5R)-4-{[(1-ethyl-1H-imidazol-5-yl)methyl]carbamoyl}-1,2-dimethyl-5-phenylpyrrolidine-2-carboxylic acid
2-(4-chlorophenyl)-4-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]morpholine
2-({[3-(4-fluorophenyl)phenyl]carbamoyl}amino)-N,N,3-trimethylbutanamide
2-(2-{1-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
1-(1-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)piperidin-4-ol
3-methyl-N-{[1-(2-phenylethyl)pyrrolidin-3-yl]methyl}pyridine-4-carboxamide
dimethyl({[(3S,4R)-4-(propan-2-yl)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidin-3-yl]sulfamoyl})amine
5-[3-(3-methoxyphenoxy)propyl]pyrimidine
N-[furan-2-yl(phenyl)methyl]-3-(1-methyl-1H-pyrazol-5-yl)propanamide
2-[(3,4-dimethoxyphenyl)methyl]-N-[2-(4-hydroxypiperidin-1-yl)ethyl]-1,3-benzoxazole-6-carboxamide
methyl 2-{1-[2-(methylamino)acetyl]-3-oxopiperazin-2-yl}acetate
7-methyl-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-(4-methyl-1H-pyrrole-2-carbonyl)piperazin-2-one
2-{2-[4-(furan-3-carbonyl)-1,4-diazepan-1-yl]-2-oxoethyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
1-ethyl-3-(oxan-4-yl)-5-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-1,2,4-triazole
1-methyl-2-(2-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)-1H-1,3-benzodiazole
(3aS,6aS)-2-(ethanesulfonyl)-5-[(1-propyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}ethyl)pyrrolidin-2-one
3-[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-1-[3-(4-methylpiperazine-1-carbonyl)phenyl]urea
(dicyclopropylmethyl)(methyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
2-(adamantan-1-ylsulfanyl)-1-(2-{[ethyl(methyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)ethan-1-one
[(4aS,8aR)-6-(2-benzyl-1,3-thiazole-4-carbonyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
(3aS,7aR)-5-methyl-2-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
(3S,9aR)-3-benzyl-8-(4-ethylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(2-ethoxypyridin-3-yl)methyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
(4aS,7aR)-1-[(3-hydroxyphenyl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione