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7-[3-(pyrimidin-2-yloxy)benzoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-{1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
4-[3-(2-fluorophenoxy)azetidine-1-carbonyl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
1-(3-fluoropyridine-4-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
methyl 2-{[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]methyl}-1,3-oxazole-4-carboxylate
(1S,5R)-3-[(4-fluoro-2-methylphenyl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]piperidine-3-carbonitrile
1-(2,2-dimethylpent-4-en-1-yl)-4-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperazine
6-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-N2,N2-diethylpyrimidine-2,4-diamine
2-(5-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
4-(5-ethylfuran-2-yl)-1-methyl-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
methyl[(3-phenyl-1,2-oxazol-5-yl)methyl]{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
N-[2-hydroxy-2-(3-phenoxyphenyl)ethyl]-2-methylpyrimidine-5-carboxamide
9-[2-(diethylamino)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-fluoro-5-[4-(3-methoxyphenyl)-3-oxopiperazine-1-carbonyl]benzonitrile
2-[2-(2,2-diphenylethyl)morpholin-4-yl]pyridine-3-carboxamide
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-4-methoxy-N-[(3S)-2-oxoazepan-3-yl]benzamide
2-{1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]pyrrolidin-2-yl}-1,3-benzothiazole
(1S,5R)-6-({3-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
N-(1,3-dihydroxy-2-methylpropan-2-yl)-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
1-(1-{[(butan-2-yl)carbamoyl]carbonyl}piperidin-4-yl)-N-(propan-2-yl)piperidine-4-carboxamide
methyl[(2E)-3-phenylprop-2-en-1-yl]{2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
2-{8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-N-(furan-2-ylmethyl)acetamide
1-(2,5-dimethylfuran-3-carbonyl)-3-[4-(methylsulfanyl)benzoyl]piperidine
(2S)-4-methyl-1-(3-phenylpropyl)-2-(propan-2-yl)piperazine
4-[(1S,2S)-2-hydroxycyclohexyl]-N-(3-phenylphenyl)piperazine-1-carboxamide
4-(1-ethyl-1H-imidazol-2-yl)-1-(1H-pyrrole-2-carbonyl)piperidine
5-{[4-(benzyloxy)piperidin-1-yl]methyl}-N-propylpyrimidin-2-amine
6-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]pyridine-3-carboxamide
1-(2-chlorophenyl)-4-(5-ethylthiophene-3-carbonyl)-5-methylpiperazin-2-one
(1S,5R)-3-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-{4-[(2E)-3-phenylprop-2-en-1-yl]morpholin-3-yl}acetamide
2-cyclopropyl-8-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(benzyloxy)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(2-methoxyphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)pyrrolidin-3-yl]methanol
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-5-phenyl-1,2-oxazole-3-carboxamide
2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-5-methyl-1H-indole
(3R,4S)-4-cyclopropyl-1-[2-(pyrrolidin-1-yl)benzoyl]pyrrolidin-3-amine
1-{2-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidine-1-carbonyl]phenyl}ethan-1-one
2-cyclopropyl-5-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]pyrimidine
(1R,5R)-6-(1H-indol-5-ylmethyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
6-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
[(4-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-oxazepan-6-yl)methyl]dimethylamine
3-(3-methylbutyl)-8-[2-(1-methylpiperidin-2-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(pyridin-3-ylmethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[(4-methylphenyl)amino]-2-phenylpropanamide
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1,3-oxazole-5-carboxamide
4-[3-({1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}oxy)benzoyl]morpholine