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N-[3-(dimethylamino)propyl]-N-methyl-1-(1,2,3,4-tetrahydroquinoline-8-carbonyl)piperidin-3-amine
2-methyl-6-(1,2,3,4-tetrahydroisoquinolin-5-yl)-2,3-dihydropyridazin-3-one
ethyl 1-[(3,4-dimethoxyphenyl)carbamoyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
6-{[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
N-{[2-methoxy-5-(1H-pyrazol-4-yl)phenyl]methyl}cycloheptanamine
3-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-5-phenyl-1,2,4-triazine
4-chloro-1-methyl-N-[3-(4-methylbenzenesulfonamido)propyl]-1H-pyrazole-5-carboxamide
1-(4-{[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}thiophen-2-yl)ethan-1-one
3-{2-[3-methyl-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-3,4-dihydroquinazolin-4-one
1-{2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]acetyl}-2-methyl-1,4-diazepan-5-one
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-4-(piperidin-1-ylmethyl)benzamide
4-sulfamoyl-N-[1-(thiophen-2-yl)propan-2-yl]benzamide
5-(3-methoxyphenoxymethyl)-N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]-1H-pyrazole-3-carboxamide
1-[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-(pyrrolidin-1-yl)benzamide
(2S,4R)-4-amino-1-(5-ethylthiophene-3-carbonyl)-N-methylpyrrolidine-2-carboxamide
5-[4-(1H-indol-3-yl)butanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
7,7-dimethyl-2-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(4aR,7aS)-1-(2-methoxyethyl)-4-[(5-methylthiophen-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-1H-imidazole
2-[(3S)-3-hydroxypyrrolidin-1-yl]-N,1-dimethyl-N-(1-methylpiperidin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
N-(2-phenylethyl)-2,8-diazaspiro[4.5]decane-2-carboxamide
6-ethoxy-3-{[4-(oxolan-2-ylmethyl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
3-{1-[(2-aminopyrimidin-5-yl)methyl]piperidin-3-yl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-[2-(pyridin-2-yl)ethyl]piperazine
N-{5-[3-(1H-pyrazol-3-yl)phenyl]quinolin-8-yl}acetamide
4-[2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-1,4-oxazepane
2-{3-[3-(benzyloxy)propyl]phenyl}-5-methyl-1,3,4-oxadiazole
2-amino-N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-4-methyl-1,3-thiazole-5-carboxamide
(3R)-1-[(8-methoxyquinolin-2-yl)methyl]pyrrolidin-3-ol
(4aR,7aS)-1-(2-methoxyacetyl)-4-(2-oxo-2-phenylacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-(2-cyclopropylpyrimidine-5-carbonyl)-1-oxa-8-azaspiro[4.6]undecane
methyl 5-[(3-hydroxy-3-methylbutan-2-yl)amino]-1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(dimethyl-1,3-thiazol-5-yl)-1-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]ethan-1-one
3-(3-fluorophenyl)-4-[2-(1H-imidazol-2-yl)benzoyl]piperazin-2-one
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxolane-3-carboxamide
N-[2-(azepan-1-yl)-2-phenylethyl]-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(2-fluorophenyl)methyl]-1-methyl-5-({[1-(morpholin-4-yl)cyclopentyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(1-{7-[(2,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
6-(2,5-dimethylphenyl)-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
2-{2-[benzyl(methyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
4-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-ylmethyl]-2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazole
1-(2,6-dimethylquinoline-4-carbonyl)-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
4-benzyl-1-methyl-3-[1-(1,3-thiazol-2-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-cyclopropyl-5-{4-[(1S,2S)-2-hydroxycyclohexyl]piperazine-1-carbonyl}-3,4-dihydropyrimidin-4-one
ethyl 4-{1-[2-(5-acetylthiophen-3-yl)acetyl]piperidin-3-yl}piperazine-1-carboxylate
N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-indole-6-carboxamide
4-phenyl-5-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}-1H-imidazole
N-{[1-(1,2,4-oxadiazol-3-ylmethyl)piperidin-3-yl]methyl}quinoline-8-sulfonamide