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8-(furan-3-carbonyl)-2-(2-methylpropyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine
(3R)-N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
9-{3H,3aH,4H,5H,9bH-cyclopenta[c]quinoline-4-carbonyl}-1,4,9-triazaspiro[5.5]undecan-5-one
(3S,4R)-1-{[cyclohexyl(methyl)carbamoyl]methyl}-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
(1R,5R)-6-methyl-3-{4-[(pyridin-2-ylsulfanyl)methyl]benzoyl}-3,6-diazabicyclo[3.2.2]nonane
N-(furan-3-ylmethyl)-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N-ethyl-5-(2-fluorophenoxymethyl)-N-(oxan-4-ylmethyl)-1H-pyrazole-3-carboxamide
9-[4-(dimethylamino)benzoyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
[(2S,6S)-4-(1H-imidazol-4-ylmethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-5-methylthiophene-2-carboxamide
2-(1,3-benzothiazol-2-yl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
methyl 3-(1H-indol-3-ylmethyl)-9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(4-{[4-(1-methyl-1,2,3,4-tetrahydroquinoline-6-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
8-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}-1-oxa-8-azaspiro[4.5]decane
1,3,6-trimethyl-N-(2-phenylpropyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3S,7S,8aS)-7-{[(2-fluoro-5-methylphenyl)methyl]amino}-3-(1H-indol-3-ylmethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
{5-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]furan-2-yl}methanol
4-cyano-N-[(3R,4S)-4-cyclopropyl-1-(pyrimidin-5-ylmethyl)pyrrolidin-3-yl]oxane-4-carboxamide
(3S,9aR)-3-benzyl-8-[(4-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(2-fluoro-5-methylphenyl)-3-{[(1R)-2-hydroxy-1-phenylethyl]amino}propanamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)acetamide
1-methyl-5-{[(2-methylphenyl)methyl]amino}-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-methyl-N4-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]pyrimidine-2,4-diamine
1-{[1-(6-methylpyridin-2-yl)-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-{[(3,4-difluorophenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
(3S,9aR)-8-(naphthalene-1-carbonyl)-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-N,N-dimethylpyrazine-2-carboxamide
(2R,6S)-4-[6-chloro-3-(piperidin-1-ylmethyl)imidazo[1,2-a]pyridine-2-carbonyl]-2,6-dimethylmorpholine
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-methyl-6-(oxolane-3-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-[({1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidin-3-yl}oxy)methyl]pyridine
3-{5-[2-(2-methyl-2,3-dihydro-1H-indol-1-yl)-2-oxoethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
5-{[4-(piperidine-1-carbonyl)piperidin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
4-(2-hydroxy-4-methylpentanoyl)-1-(2-methoxyphenyl)piperazin-2-one
3-{1-[(6-chloro-2H-chromen-3-yl)methyl]piperidin-3-yl}-N-(2-fluorophenyl)propanamide
4-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methoxyquinoline
N-(2-methoxyethyl)-5-[4-(methylsulfamoyl)phenyl]furan-2-carboxamide
3-[(dimethylamino)methyl]-1-{3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}piperidin-3-ol
ethyl 5-{[2-(benzylsulfanyl)ethyl]carbamoyl}-1H-imidazole-4-carboxylate
N-[(3R,4S)-4-propyl-1-(trimethylpyrimidin-4-yl)pyrrolidin-3-yl]methanesulfonamide
5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]-1-[2-(pyridin-2-yl)ethyl]piperidin-2-one
2-ethyl-5-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
3-(1H-imidazol-2-yl)-N-methyl-N-[2-(phenylsulfanyl)ethyl]benzamide
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-2-methyl-1,3-thiazole-4-carboxamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl})amine
1-{3-tert-butyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methylpropan-1-one
{2-[3-(2-methylphenoxymethyl)piperidin-1-yl]quinolin-3-yl}methanol
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]acetamide
6,7-dimethoxy-3-(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-3,4-dihydroquinazolin-4-one