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2-({[2-(3-methylphenyl)-1,3-thiazol-4-yl]methyl}amino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[1-(4-fluorobenzoyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
1-[4-(2-cyclobutyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]-3-hydroxy-2-phenylpropan-1-one
5-[(4-hydroxypiperidin-1-yl)methyl]-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,2-oxazole-3-carboxamide
N-[(2-methoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)-3-(1H-1,2,4-triazol-1-yl)propanamide
(4aS,8aS)-2-({2-[(2-methylphenyl)methoxy]phenyl}methyl)-decahydro-2,7-naphthyridin-4a-ol
3-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-1-[4-(1H-pyrazol-1-yl)phenyl]urea
3-(2-fluorophenyl)-3-phenyl-N-[2-(1H-pyrazol-1-yl)ethyl]propanamide
2-(dimethylamino)-N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)benzamide
3-[(3S,4R)-1-benzyl-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-N-cyclooctylpropanamide
8-[(3,4-dimethoxyphenyl)methyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-[(2S,4R)-1-[(2,5-dimethylphenyl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
6-(2-chlorophenyl)-N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-(2,5-dioxoimidazolidin-4-yl)propanamide
N-[(3-chlorophenyl)methyl]-N-cyclopropyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-4-methylphenol
2-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperidine-3-carbonyl)pyridine
3-[(carbamoylmethyl)sulfamoyl]-N-[(1-propyl-1H-pyrazol-4-yl)methyl]benzamide
5-oxo-1-({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)pyrrolidine-3-carboxylic acid
(4aS,7aR)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(dimethylsulfamoyl)-N-(2-methyl-1-benzofuran-5-yl)piperazine-1-carboxamide
4-{[5-(3-methanesulfonylphenyl)-1,2,4-oxadiazol-3-yl]methyl}-1-methylpiperidine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
4-[5-(1-benzylpiperidin-2-yl)-3-methyl-1H-1,2,4-triazol-1-yl]-2-methylpyridine
dimethyl({[5-(6-phenylpyridazin-3-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl})amine
N,N-dimethyl-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine-4-sulfonamide
1-[1-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-2-ol
3-(benzylamino)-N-[(1S)-1-phenylethyl]-5-[(propan-2-yl)sulfamoyl]benzamide
(1S,6R)-9-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
4-(3-hydroxy-3-methylbutyl)-N-[3-(3-oxopiperazin-1-yl)propyl]benzamide
8-(4-methyl-1,3-thiazole-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
9-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-2-[3-(dimethylamino)propyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
8-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
[(3R,4S)-4-(morpholin-4-ylmethyl)-1-[(2-phenylphenyl)methyl]pyrrolidin-3-yl]methanol
3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-one
N-(3-hydroxypropyl)-1,5-dimethyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
ethyl 4-(6-methyl-3-{[(2-phenylethyl)amino]methyl}quinolin-2-yl)piperazine-1-carboxylate
3-(2-methylpropyl)-5-[(phenylsulfanyl)methyl]-1H-1,2,4-triazole
N-(1-{1-[(2,4-difluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methylbenzamide
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyridin-4-amine
N-cyclopentyl-3-(4-methyl-5-oxo-1,4-diazepane-1-carbonyl)benzene-1-sulfonamide
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
3-hydroxy-1-(2-methoxyethyl)-3-{[(1,2-oxazol-3-ylmethyl)amino]methyl}piperidin-2-one
2-(4-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)ethan-1-ol
5-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
2-(4-methoxy-3,5-dimethylphenyl)-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]acetic acid
N-cyclopropyl-4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]piperazine-2-carboxamide
8-[(1-ethyl-1H-indol-4-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid