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1-(2-chlorophenyl)-3-[1-(1-cyclohexylpiperidin-4-yl)-1H-pyrazol-5-yl]urea
4-(2,6-dimethylphenyl)-6-methylpyrimidin-2-amine
[(2R)-1-{[2-(4-chlorophenyl)-7-methoxyquinolin-3-yl]methyl}pyrrolidin-2-yl]methanol
3-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-N-benzyl-N-methylpropanamide
4-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-5,6-dimethylpyrimidine
3-ethyl-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-methyl-N-[1-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)pentyl]thiophene-2-carboxamide
2-[3-(2-methylphenoxy)azetidin-1-yl]pyrimidin-4-amine
8-oxo-7-(prop-2-en-1-yl)-N-[(3S)-pyrrolidin-3-yl]-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
5-methyl-5-phenyl-1-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}piperidin-2-one
2-(2-oxopyrrolidin-1-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[1-(2-hydroxy-2-phenylethyl)-4-phenyl-1H-imidazol-5-yl]benzonitrile
1-(1-benzylpiperidin-4-yl)-N-[2-(1H-imidazol-4-yl)ethyl]piperidine-3-carboxamide
(2S,4R)-4-amino-N,N-diethyl-1-(1H-1,2,4-triazole-5-carbonyl)pyrrolidine-2-carboxamide
[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
(3S,9aR)-3-(4-aminobutyl)-8-(3,5-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(3R,7S,8aS)-3-[(benzylsulfanyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,5-difluorobenzamide
4-(hydroxymethyl)-1-{[5-(1,2-oxazol-5-yl)thiophen-2-yl]sulfonyl}azepan-4-ol
N-cyclopropyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
2-cyclohexyl-N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-1,3-benzoxazole-6-carboxamide
1-(1H-imidazole-5-carbonyl)-4-[2-(morpholin-4-yl)ethyl]-1,4-diazepan-6-ol
(1R,3S)-3-(2-hydroxyethoxy)-7-[(3E)-4-methylhex-3-en-1-yl]-7-azaspiro[3.5]nonan-1-ol
N-(cyclohexylmethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
methyl 4-{[(1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}piperidin-4-yl)amino]methyl}benzoate
N-{[1-(3,3,3-trifluoropropyl)pyrrolidin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
4-({3-[2-(hydroxymethyl)piperidin-1-yl]propyl}carbamoyl)benzoic acid
N-(4-{[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}phenyl)cyclopropanecarboxamide
N-[4-(2-methanesulfonylacetamido)-2-methoxyphenyl]butanamide
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-2,3-dihydro-1-benzothiophene-2-carboxamide
3-{5-[(2-phenylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
6-(methoxymethyl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyridine-2-carboxamide
1-(pyrazine-2-carbonyl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidin-4-amine
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-5-(4-methoxyphenyl)-N-methyl-1,2,4-triazin-3-amine
6-({3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{5-[3-(2-phenylethyl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
[5-({4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)furan-2-yl]methanol
1-[4-(morpholine-4-carbonyl)benzenesulfonyl]pyrrolidine-2-carboxylic acid
1-{4-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
8-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
1-[benzyl(methyl)amino]-3-[5-({[3-(dimethylamino)-2,2-dimethylpropyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
methyl 1-[(3R,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-[(3-methoxyphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-[7-(3-methoxypiperidine-1-carbonyl)-1-(2-phenylethyl)-1H-1,3-benzodiazol-5-yl]methanesulfonamide
5-[2-(ethylamino)ethyl]-1-[2-(propan-2-yloxy)ethyl]pyrrolidin-2-one
(1R,5S,8R)-3-({3-[(4-ethylpiperazin-1-yl)methyl]-2,5-dimethylphenyl}methyl)-3-azabicyclo[3.2.1]octan-8-ol
N-(1,2-oxazol-3-ylmethyl)-4-(1H-pyrazol-3-yl)benzamide
4-{[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]methyl}-1λ6-thiane-1,1-dione
3-[(1-ethylpiperidin-2-yl)methyl]-3H,4H-pyrido[4,3-d]pyrimidin-4-one
N-[2-(5-methylfuran-2-yl)phenyl]-3-(1H-pyrazol-3-yl)piperidine-1-carboxamide
1-(5-ethyl-1,2,4-oxadiazol-3-yl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine