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3-benzyl-1-(2-chlorophenyl)-4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(oxolan-2-ylmethyl)-3-(1H-pyrazol-1-ylmethyl)-N-(thiophen-3-ylmethyl)benzamide
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-1-methylazepane-2-carboxamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(pyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(2-ethyl-1H-imidazol-1-yl)-1-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
methyl 2-{[1-(cyclohexylmethyl)-3-(methylcarbamoyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}acetate
2-({2-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N,2,8-trimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]quinoline-4-carboxamide
(2S)-N2-[2-(4-fluorophenyl)ethyl]-N2-(pyridin-3-ylmethyl)pyrrolidine-1,2-dicarboxamide
2-[2-(1-methylpiperidin-2-yl)ethyl]-2,3-dihydro-1,2-benzothiazol-3-one
4-(7-chloro-1-methyl-1H-indole-2-carbonyl)-3-(2-hydroxyethyl)piperazin-2-one
6-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}-N-[4-(1H-pyrazol-1-yl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
2-[(4-chlorophenyl)methyl]-8-(furan-3-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
[2-(1H-imidazol-4-yl)ethyl]({[2-(propylsulfanyl)pyrimidin-5-yl]methyl})amine
ethyl 4-[4-benzyl-6-(cyclopropylmethoxy)-3-oxo-1,4-diazepan-1-yl]piperidine-1-carboxylate
2-(dimethylamino)-2-(2-fluorophenyl)-N-[2-(pyridin-3-yl)ethyl]acetamide
(3S,4S)-4-cyclopropyl-1-[2-(1H-indazol-1-yl)acetyl]pyrrolidine-3-carboxylic acid
1-[(6-chloropyridin-2-yl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(2-hydroxyethyl)-8-[3-(4-methylphenyl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
4-[(2S,3S)-2-amino-3-methylpentanoyl]-1-(2-methylphenyl)piperazin-2-one
1-cyclohexyl-4-[3-(1H-imidazol-2-yl)imidazo[1,2-a]pyridine-2-carbonyl]piperazine
6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-4-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-1,4-diazepan-2-one
N-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-2-methyl-N-(oxolan-2-ylmethyl)propanamide
5,6-dimethyl-N4-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}pyrimidine-2,4-diamine
1-[(1s,4s)-4-aminocyclohexyl]-N-[2-(1,3-thiazol-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}morpholine
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}oxolane-3-carboxamide
4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-N-(2,4,6-trimethylphenyl)piperidine-1-carboxamide
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)cyclopropane-1-carboxamide
N-{2-methyl-1-[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]-1-oxopropan-2-yl}thiophene-2-carboxamide
(3S,4R)-1-{4-methyl-3-oxo-1H,2H,3H-pyrazolo[3,4-b]pyridine-6-carbonyl}-4-phenylpyrrolidine-3-carboxylic acid
1-(methoxymethyl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]cyclobutane-1-carboxamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2,3-dimethylquinoxaline-6-carboxamide
4-({2-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)piperazin-2-one
N-[3-({[1-(2,4-dimethylphenyl)ethyl]carbamoyl}methoxy)phenyl]propanamide
1-(5-ethyl-2-methylpyrimidin-4-yl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]piperidin-4-amine
1-[5-methoxy-2-({[3-(pyridin-3-yl)propyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
1-[(2,5-dimethoxyphenyl)methyl]-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazine
5-butyl-1'-(6-methylpyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-{1-[2-amino-6-methyl-5-(prop-2-en-1-yl)pyrimidin-4-yl]piperidin-4-yl}-1,3-oxazolidin-2-one
(3S,7S,8aS)-7-{[(3-fluorophenyl)methyl]amino}-3-[(1R)-1-hydroxyethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
N-methyl-N-(pentan-3-yl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-[(2E)-2-methylpent-2-en-1-yl]-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-[3-(2-methyl-1H-imidazol-1-yl)propyl]piperidine
1-(2-ethoxypyridine-3-carbonyl)-2-(pyrrolidine-1-carbonyl)piperazine
1-[3-(2-methyl-1H-imidazol-1-yl)propyl]-4-(6-methylpyridin-2-yl)piperazine
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-methyl-6-(pyrazine-2-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one