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4-methoxy-N-(oxolan-3-ylmethyl)-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
3-phenyl-6-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyridazine
2-butyl-N-[(4-methoxyphenyl)methyl]-4-methyl-3-oxopiperazine-1-carboxamide
2-{1-cyclopentyl-4-[(4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[(5-{[3-(2-aminoethyl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]-3,3-dimethylurea
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-3-(2-phenylethyl)piperidine-3-carboxylic acid
5-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-hexyl-8-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
3-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](methyl)[2-(1H-pyrazol-1-yl)ethyl]amine
5-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-4-phenyl-1H-imidazole
N-methyl-2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-(1H-pyrazol-5-ylmethyl)acetamide
2-methyl-2-(2-{[1-(6-methylpyridin-2-yl)ethyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)propanoic acid
4-{[(3R)-3-hydroxypyrrolidin-1-yl]sulfonyl}-N-(1H-imidazol-2-ylmethyl)benzamide
1-methyl-6-(1H-pyrazol-3-ylmethyl)-3-[4-(trifluoromethoxy)phenyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-(1-cycloheptylpiperidin-3-yl)-3-(1,2-oxazinan-2-yl)propanamide
2-(azepan-1-yl)-N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
N-[1-(furan-2-ylmethyl)piperidin-4-yl]-2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetamide
6-(methoxymethyl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyrimidin-4-amine
N-(5-{[1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}thiophen-2-yl)acetamide
1-[(3S,4S)-3-hydroxy-4-[(2-methoxyethyl)(methyl)amino]pyrrolidin-1-yl]-4-(1H-indol-3-yl)butan-1-one
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]acetamide
2-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-N-(2-phenylethyl)acetamide
1-(4-chlorophenyl)-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)cyclopropane-1-carboxamide
1-butyl-5-[(2,3,4-trifluorophenyl)methyl]-1H-1,2,4-triazole
(2S,4S)-4-amino-1-{2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetyl}-N-methylpyrrolidine-2-carboxamide
1-(benzenesulfonyl)-4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperazine
8-(6-oxopiperidine-3-carbonyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-hydroxy-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]acetamide
N-[(3R,4S)-4-cyclopropyl-1-(1-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)pyrrolidin-3-yl]methanesulfonamide
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-4-phenylbutane-1,4-dione
N-(1H-indazol-6-yl)morpholine-4-carboxamide
N-(1-{2-[3-(morpholine-4-carbonyl)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-phenoxyacetamide
methyl 3-{[(3-methoxyphenyl)formamido]methyl}-5-[3-(trifluoromethyl)benzamido]benzoate
1-[3-(difluoromethoxy)benzoyl]-3-propylpiperidine-3-carboxylic acid
5-cyclobutyl-1-(2-hydroxyethyl)-N-(1-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(7-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
3-ethyl-8-[(3-methoxyphenyl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(dimethylamino)ethyl]-1-methyl-N-[(3-methylthiophen-2-yl)methyl]-1H-pyrazole-5-carboxamide
N-(2,4-dimethoxyphenyl)-3-(6-methoxynaphthalene-2-carbonyl)piperidine-1-carboxamide
N-[2-(3-hydroxy-4-methoxyphenyl)ethyl]-3-(2-methyl-1H-indol-1-yl)propanamide
2-cyclopropyl-5-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]pyrimidine
2-(3-methoxypropyl)-8-(2-phenoxypropanoyl)-2,8-diazaspiro[4.5]decan-3-one
methyl[3-(5-methylfuran-2-yl)butyl]{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(oxane-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(2H-1,3-benzodioxol-4-ylmethyl)(methyl)[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]amine
8-(2-fluorobenzoyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-[2-(diethylamino)ethyl]-6-phenyl-2-(pyrrolidin-1-yl)pyridine-3-carboxamide
2-ethyl-5-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]pyrimidine