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N-[1-(methoxymethyl)cyclopentyl]-2,5-dimethyl-1,3-thiazole-4-carboxamide
2-ethoxy-5-{2-[(2-hydroxybutyl)amino]pyrimidin-4-yl}benzoic acid
(1R,5R)-6-(2-methoxyethyl)-3-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonane
3-methyl-N-(4-methyl-1,3-thiazol-2-yl)-1H-1,2,4-triazole-5-carboxamide
2-butyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,3-benzoxazole-5-carboxamide
3-methoxy-5-methyl-N-[1-methyl-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]thiophene-2-carboxamide
1-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}-2-(2-phenylethyl)pyrrolidine
2-{1-[2-(dimethylamino)-4-methylpyrimidin-5-yl]-N-methylformamido}-2-(pyridin-3-yl)acetic acid
ethyl 5-(2,3-dihydroxypropyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
5-{[(3,5-difluorophenyl)methyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{2-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]ethyl}-2,2-dimethylpropanamide
1-cyclopropyl-3-{2-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,2-oxazole-3-carbonyl)piperidine
N-[(2-methoxynaphthalen-1-yl)methyl]-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
9-(3-fluoropyridine-2-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-cyclohexyl-N-(cyclopropylmethyl)-N-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(3aR,5R,6S,7aS)-2-[8-(trifluoromethyl)quinolin-4-yl]-octahydro-1H-isoindole-5,6-diol
1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
3-(dimethyl-1,2-oxazol-4-yl)-1-[2-(4-methylpentyl)morpholin-4-yl]propan-1-one
2,5-dimethyl-3-(4-{[5-(oxan-2-yl)furan-2-yl]methyl}piperazin-1-yl)pyrazine
N-[(3R,4R)-3-hydroxy-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-4-yl]pyridine-2-carboxamide
1-(2-methoxyethyl)-3-methyl-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-methyl-1H-pyrazole-5-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-(1-{[1-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)acetamide
7-(5-hydroxy-1,2-dimethyl-1H-indole-3-carbonyl)-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(1,1-dioxo-1λ6-thiomorpholin-4-yl)-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}benzamide
3-[(3S,4R)-1-benzyl-4-(4-methylpiperazin-1-yl)piperidin-3-yl]-N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methylpropanamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
5-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(3R,5S)-N3-(4-fluorophenyl)-N5-(naphthalen-1-ylmethyl)-1-(pyridin-4-ylmethyl)piperidine-3,5-dicarboxamide
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-(4-methyl-3-phenyl-1H-pyrazol-1-yl)acetamide
N'-(5-chloro-2-methylphenyl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]propanediamide
3-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]benzene-1-sulfonamide
(1S,6R)-9-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3,9-diazabicyclo[4.2.1]nonan-4-one
6-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N2,N2-diethylpyrimidine-2,4-diamine
5-methyl-3-{6-methylthieno[2,3-d]pyrimidin-4-yl}-1H-indole
3-(4-hydroxyphenyl)-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
2-[4-({4-[(4-chlorophenyl)methyl]piperazin-1-yl}methyl)-3-methyl-1H-pyrazol-1-yl]ethan-1-ol
N'-(3,5-dimethylphenyl)-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methylpropanediamide
N-[2-(morpholin-4-yl)ethyl]-4-(4-{[2-(thiophen-2-yl)ethyl]amino}piperidin-1-yl)benzamide
4-(4-methoxyphenyl)-N-(oxolan-3-yl)butanamide
6-chloro-3-({3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}methyl)-4H-chromen-4-one
N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
2-[(3R,4S)-3-(3-methoxy-5-methylthiophene-2-amido)-4-propylpyrrolidin-1-yl]acetic acid
N-[(1-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}piperidin-3-yl)methyl]-3-phenylpropanamide
7-[(2-fluorophenyl)methyl]-2-[3-(methylsulfanyl)propyl]-2,7-diazaspiro[4.5]decan-6-one
(2S,4R)-4-(furan-3-amido)-N-methyl-1-(2-phenoxyethyl)pyrrolidine-2-carboxamide
3-(2-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-2-yl}ethyl)phenol
5-(azepane-1-carbonyl)-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[3-(2-phenylethyl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one