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1-butyl-4-[2-(4-fluoropiperidin-1-yl)-2-oxo-1-phenylethyl]piperazine-2,3-dione
methyl (2S,4S,5R)-1,2-dimethyl-5-(2-methylphenyl)-4-(4-methylpiperazine-1-carbonyl)pyrrolidine-2-carboxylate
N-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
1-methyl-4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydroquinolin-2-one
1-(2-methylpropyl)-4-[4-(naphthalen-2-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
N-cyclohexyl-N-[2-(3,4-dimethoxyphenyl)ethyl]oxolane-3-carboxamide
(1S,5R)-3-cyclobutanecarbonyl-N-(2,4-dimethylphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
9-(6-methyl-2-propylpyrimidin-4-yl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
N4-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-[(3R,4S)-4-(3-methoxyphenyl)-1-methylpyrrolidin-3-yl]cyclopentanecarboxamide
5-{2-methylpyrido[2,3-d]pyrimidin-4-yl}-3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(2S,4R)-4-amino-1-{[2-(ethylamino)pyrimidin-5-yl]methyl}-N-methylpyrrolidine-2-carboxamide
ethyl 1-(cyclopropylmethyl)-5-[2-(morpholin-4-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-{1-[7-(1H-indole-6-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}-3,5-dimethylbenzamide
3-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,2-oxazole
(4aR,7aS)-1-(pyrimidin-2-yl)-4-[2-(1H-1,2,4-triazol-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)carbamoyl]pyridin-1-ium-1-olate
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-(4-methylbenzoyl)piperazin-2-yl}ethan-1-ol
4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazine-1-sulfonamide
4-{[3-(2-chlorophenoxy)azetidin-1-yl]methyl}-5-methyl-1-propyl-1H-pyrazole
8-acetyl-2-(1H-imidazol-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-[3-(3-methylphenyl)piperidin-1-yl]pyrazine
ethyl 3-[(2E)-3-phenylprop-2-en-1-yl]-1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidine-3-carboxylate
1-[(3-methylphenyl)methyl]-4-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanoyl}piperazin-2-one
[3-(cyclopropylmethyl)-1-(2,3-difluoro-6-methoxybenzoyl)piperidin-3-yl]methanol
3-(1-methylpiperidin-2-yl)-1-[3-(1H-pyrazol-1-yl)azetidin-1-yl]propan-1-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(2-oxopyrrolidin-1-yl)propanamide
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(ethanesulfonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-(furan-2-yl)propan-1-one
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(1-phenoxypropan-2-yl)piperidin-4-yl]propanamide
1-(2-benzylmorpholin-4-yl)-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]ethan-1-one
N-{[1-(3,5-dimethylphenyl)cyclopentyl]methyl}-2,7-dioxo-1,3-diazepane-4-carboxamide
4-(methoxymethyl)-5-methyl-N-[(4-sulfamoylphenyl)methyl]-1,2-oxazole-3-carboxamide
4-(1-{[6-(dimethylamino)pyridin-3-yl]methyl}piperidin-3-yl)benzoic acid
3-(2-methylpropyl)-1-(2-phenylethyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
[(2-ethoxyphenyl)methyl](ethyl)(pyridin-3-ylmethyl)amine
N-cyclopentyl-1-methyl-5-[(1-methyl-1H-indol-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-(4-methoxypiperidin-1-yl)-N-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-(2-methoxyphenoxy)-1-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propan-1-one
2-[(4aR,7aS)-4-{[3-(2-aminoethyl)phenyl]methyl}-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
(1R,2S,6R,7S)-4-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-azatricyclo[5.2.2.02,6]undecane
N-cyclopropyl-3-oxo-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopentane-1-carboxamide
1-(1-{1-[2-(azepan-1-ylmethyl)-2-methylpropyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-ol
(1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methanol
1-[(furan-2-ylmethyl)carbamoyl]-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
3,5-dimethoxy-2-{[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]methyl}benzoic acid
8-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one