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2-[methyl(pyridin-4-ylmethyl)amino]-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1,3-dimethyl-N-(1,2-oxazol-3-ylmethyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-[(4-amino-6-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}pyrimidin-2-yl)sulfanyl]-N,N-dimethylacetamide
1-{2-[1-(1,4-dimethyl-1H-indole-2-carbonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
1-[(1-ethylpiperidin-3-yl)methyl]-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
6-{[(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)amino]methyl}-1,4-oxazepan-6-ol
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[4-(dimethylamino)phenyl]ethan-1-one
(2S,4S)-4-amino-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1-methylpyrrolidine-2-carboxamide
7-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-2-oxa-7-azaspiro[4.5]decane
N-[1-(2,5-dimethylphenyl)ethyl]-2-ethoxyacetamide
(2S,4R)-N-ethyl-4-{4-[4-(pyrrolidin-1-ylmethyl)phenyl]-1H-1,2,3-triazol-1-yl}pyrrolidine-2-carboxamide
1-(2-methoxy-5-{[(2-phenoxyethyl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
N-(4-{2-[3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethoxy}phenyl)propanamide
1-(furan-3-carbonyl)-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
1-(pyridin-4-yl)-4-[(2,4,5-trimethylphenyl)methyl]piperazine
N-cyclohexyl-2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-methyl-1,3-oxazole-4-carboxamide
1-(3-{[4-(ethylamino)pyrimidin-2-yl]amino}propyl)pyrrolidin-2-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(1H-imidazol-1-yl)acetamide
3,5-dichloro-4-methyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]benzamide
3-methyl-7-[6-(piperidin-1-yl)pyrimidin-4-yl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
methyl (2S)-4-methyl-2-({5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazol-3-yl}formamido)pentanoate
3-methyl-1-[7-(1-methyl-1H-pyrrole-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidine
(3R,4R)-4-{[6-(4-fluorophenyl)pyridazin-3-yl]amino}piperidin-3-ol
5-benzyl-4-[2-(dimethylamino)acetyl]-1-(4-methylphenyl)piperazin-2-one
(1r,4r)-4-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)cyclohexan-1-ol
2-(4-chlorophenoxy)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
1-benzyl-N,N-dimethyl-5-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(3-methoxyphenyl)-1-{2-[2-(pyridin-2-ylsulfanyl)acetamido]ethyl}-1H-1,2,3-triazole-4-carboxamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
methyl 6-{[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}pyridine-2-carboxylate
4-[(2,3-dimethoxyphenyl)methyl]-3-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]piperazin-2-one
3,5-dimethyl-N-(3-methyl-1-{7-[(6-methylpyridin-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)benzamide
5-(ethanesulfonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(furan-2-ylmethyl)propanamide
4-[(6-methoxy-1H-indazol-3-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
2-{4-[(2,4-difluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-(dimethylamino)propan-2-ol
4-(1H-pyrazol-3-yl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]benzamide
N-[2-methyl-2-(morpholin-4-yl)propyl]-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
(1R,5R)-6-[(5-methylthiophen-2-yl)methyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
(1R,6S)-N-[5-methoxy-2-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
2-amino-6-(2,4-dimethoxyphenyl)-4-(2-ethylpyrimidin-5-yl)pyridine-3-carbonitrile
(1S,6R)-9-[4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-methyl-N-{1-[7-(3-methylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}propanamide
2-methyl-1-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1,4-dihydroquinolin-4-one
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl](propan-2-yl)amine
3-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
4-(4-fluorophenoxy)-1-[4-(1H-imidazol-1-yl)benzoyl]piperidine
(3S,9aR)-8-(3,5-dichlorobenzoyl)-3-[(4-hydroxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-methyl-N-(1,2-oxazol-3-ylmethyl)-1-[3-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
N-(1-{1-[(2,4-dimethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide