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1-(1,1-dioxo-1λ6-thiolan-3-yl)-N-[(2-methoxyphenyl)methyl]piperidine-4-carboxamide
3-{2-[1-(2-aminopyridine-4-carbonyl)piperidin-2-yl]ethyl}phenol
4-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
2-[(3S)-3-hydroxypyrrolidine-1-carbonyl]-7-(prop-2-en-1-yl)-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
5-{1-[5-(3,5-dimethylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole
1-amino-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)cyclopropane-1-carboxamide
1-{[2-(furan-2-yl)phenyl]methyl}piperidin-4-amine
(3S,4S)-4-methyl-1-[4-(1,3-oxazol-5-yl)benzoyl]piperidine-3,4-diol
2-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(2-methylfuran-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-benzyl-5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}pyrimidin-2-amine
1-{5-[(5-methylfuran-2-yl)methyl]-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-1,4-diazepan-5-one
2-tert-butyl-N-(2-chloropyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
3-ethyl-1-(2-phenylethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[4-(3-methyl-5-propyl-1-benzofuran-2-carbonyl)piperazin-1-yl]propanamide
2-methyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N3-[(4,6-dimethylpyridin-3-yl)methyl]piperidine-1,3-dicarboxamide
N-(1-{7-[(3,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
1-(1-methyl-1H-pyrrole-2-carbonyl)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
4,6-dimethyl-2-[9-oxo-8-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carbonitrile
3-(3-fluorophenyl)-5-{spiro[2.4]heptane-1-carbonyl}-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-{4-[3-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}-N-methyl-6-[4-(methylsulfanyl)phenyl]-N-(1,2-oxazol-3-ylmethyl)pyridine-3-carboxamide
N-benzyl-6-(4-ethylpiperazin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-cyclopentyl-4-[6-(morpholin-4-yl)pyrimidin-4-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
5-{3-[1-(but-3-en-1-yl)-1H-pyrazol-3-yl]phenyl}pyrimidine
2-(dimethyl-1,2-oxazol-4-yl)-N-(5-methyl-2,1,3-benzothiadiazol-4-yl)pyrrolidine-1-carboxamide
(2E)-1-[(4aR,8aS)-6-(5-acetylthiophene-3-carbonyl)-decahydro-1,6-naphthyridin-1-yl]-3-(4-fluorophenyl)prop-2-en-1-one
(1R,5R)-6-(2,3-dimethyl-1H-indole-7-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-{2-[4-(2-methylpropyl)morpholin-2-yl]ethyl}-1H-pyrrole-2-carboxamide
(2R)-N-[6-(3-methoxyphenoxy)pyridin-3-yl]-2-methylpiperazine-1-carboxamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]acetamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-(pyrrolidin-1-yl)propanamide
2-(4-methylphenyl)-N-[2-(1H-1,2,4-triazol-1-yl)ethyl]quinoline-4-carboxamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)propane-1-sulfonamide
4-(4-chloro-1-methyl-1H-indazol-3-yl)-3-cyclobutyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-(5-phenoxyfuran-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
2-(2-methoxyethyl)-6-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1,3-benzoxazole
1-cycloheptanecarbonyl-3-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
1-[4-(1H-imidazol-1-yl)butanoyl]-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-[2-(methylsulfanyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2R,3R)-3-{[2-(3-fluorophenyl)ethyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(3R,4R)-1-[(5-chlorothiophen-2-yl)methyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
N-methyl-3-(5-methylthiophen-2-yl)-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
N-[4-(2,2-dimethylpropanamido)-3-methylphenyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
2-(5-ethyl-1H-pyrrole-2-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-(3-methoxypropyl)-9-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
3-(3-fluorophenyl)-6-(1-methyl-1H-pyrazole-5-carbonyl)-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(4aR,7aS)-1-(2-methylpropyl)-4-[(1-propyl-1H-imidazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione