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(4aR,7aS)-1-cyclobutanecarbonyl-4-[3-(pyridin-3-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidin-4-yl)pyridine
{2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-1,3-thiazol-4-yl}methanol
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2-methoxyphenyl)methyl]piperidine
3-(2-amino-1,3-thiazol-4-yl)-1-(6,7-dimethoxy-1-methyl-1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
4-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-(2-methylpropyl)pyrrolidin-2-one
(1R,2R,6S,7S)-4-[(5-methoxy-1H-indazol-3-yl)methyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
1-[(2,6-dichlorophenyl)methyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
4-(2,4-difluoro-3-methoxyphenyl)-1-(2-methanesulfonylethyl)-1H-1,2,3-triazole
(2S,3S)-3-methyl-2-({2-methylimidazo[1,2-a]pyrimidin-3-yl}formamido)pentanamide
2-(furan-2-yl)-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-2-oxoacetamide
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-5-propyl-1,2-oxazole-3-carboxamide
(3R,5S)-5-(3-fluorophenoxymethyl)-1-[(4-hydroxyphenyl)methyl]-N-[2-(1H-imidazol-4-yl)ethyl]piperidine-3-carboxamide
N-[(7-chloro-4-{[(4-fluorophenyl)methyl]amino}quinazolin-2-yl)methyl]propane-1-sulfonamide
4-methoxy-N-{[1-(thian-4-yl)piperidin-3-yl]methyl}benzene-1-sulfonamide
4-{[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(4-fluorophenyl)ethyl)piperidin-1-yl]methyl}phenol
4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]pyrimidin-2-amine
1-[4-chloro-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-3-ethylpiperidine-3-carboxylic acid
2-(oxolan-2-ylmethyl)-9-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(4aS,7aR)-N,N-dimethyl-4-[(4-methyl-1H-imidazol-5-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-sulfonamide
5-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-N-methyl-N-[1-(pyridin-2-yl)ethyl]-1H-pyrazole-3-carboxamide
{1-[4-(furan-2-yl)benzoyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
4-(furan-3-carbonyl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
N-butyl-4-{[(1-methylpiperidin-2-yl)methyl]amino}pyridine-2-carboxamide
1-cyclohexyl-N-[(1S,2R)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-yl]piperidine-4-carboxamide
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(4-chlorophenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
5-[(3-fluorophenyl)methyl]-3-(3-fluoropropyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
4-oxo-4-[2-(trifluoromethyl)morpholin-4-yl]butane-1-sulfonamide
3-{1-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]piperidin-3-yl}benzoic acid
N-[2-(3,4-dimethoxyphenyl)ethyl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
6-chloro-4-[4-(propan-2-yl)piperazine-1-carbonyl]-2-(1H-pyrazol-4-yl)quinoline
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]propan-1-one
2-(methoxymethyl)-1-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidine
3-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl](oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
2-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-ethyl-5-methyl-1H-pyrazole-4-sulfonamide
2-[1-(5-fluoro-1H-indole-2-carbonyl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
5-({[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]amino}methyl)-N-methylfuran-2-carboxamide
1-{[3-(3-fluorophenyl)oxolan-3-yl]methyl}-4-(pyridin-3-ylmethyl)-1,4-diazepane
3-{1-[2-(diethylamino)acetyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
1,3-dimethyl-5-{2-oxo-2-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethyl}imidazolidine-2,4-dione
2-methoxy-1-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methylpropan-1-one
N-(1-benzothiophen-2-ylmethyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(2E)-3-(furan-2-yl)prop-2-enoyl]piperidin-4-yl}oxy)benzamide
(1R,2R,6S,7S)-4-(4-methyl-5-phenylthiophene-2-carbonyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
N-[(4-chlorophenyl)methyl]-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-propylacetamide
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N,2,5,6-tetramethylpyrimidin-4-amine