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N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-[(1S,2R)-2-(tert-butylcarbamoyl)cyclohexanecarbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
(4-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}phenyl)methanol
4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine-1-sulfonamide
5-{1-[(2,4-difluorophenyl)methyl]piperidin-4-yl}-3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]imidazolidine-2,4-dione
(1R,7S)-3-(2-ethoxyethyl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(1R)-2-{3-[3-(3-methoxypyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}-1-phenylethan-1-ol
2-cyclopropanecarbonyl-8-[(3,4-dimethylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-{1-[(2-fluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(2-methoxyphenyl)-1-benzofuran-2-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-[3-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]urea
[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl](methyl)(pyrazin-2-ylmethyl)amine
1-({[1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}methyl)cyclohexan-1-ol
2-amino-4-(1-ethyl-1H-pyrazol-4-yl)-6-(thiophen-2-yl)pyridine-3-carbonitrile
(1R,5S)-8-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-3,8-diazabicyclo[3.2.1]octane
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-one
1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
6-[1-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)piperidin-4-yl]pyrimidin-4-ol
N2-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-N1-(3-methylpyridin-2-yl)ethane-1,2-diamine
(2E)-N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(pyridin-2-yl)prop-2-enamide
4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1-(3-propyl-1H-pyrazole-5-carbonyl)piperidine
4-(hydroxymethyl)-3-[2-(naphthalen-1-yl)ethyl]-1,3-oxazolidin-2-one
N4-methyl-N2-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrimidine-2,4-diamine
N-(1-{4-[(dicyclopropylmethyl)(methyl)carbamoyl]phenyl}-1H-pyrazol-4-yl)furan-3-carboxamide
3-(3-oxo-3-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}propyl)-3,4-dihydroquinazolin-4-one
7-(1,3-benzothiazol-2-yl)-4-[(2-fluoro-4-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-{4-[methyl(oxolan-3-yl)amino]piperidin-1-yl}benzamide
2-(4-{[(dimethyl-1,2-oxazol-4-yl)methyl]amino}-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)acetic acid
2-[2-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
2-methyl-N-(1,4-oxazepan-6-ylmethyl)-1,3-benzothiazole-6-sulfonamide
ethyl 4-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-amido}piperidine-1-carboxylate
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl][(1-cyclopentylpiperidin-4-yl)methyl](pyridin-3-ylmethyl)amine
8-methoxy-3-[(2-methylpyridin-4-yl)methyl]-3,4-dihydroquinazolin-4-one
2-(dimethylamino)-N-{5-[({[1-(hydroxymethyl)cyclobutyl]methyl}(methyl)carbamoyl)amino]-2-methylphenyl}acetamide
4,4,4-trifluoro-1-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)butan-1-one
N-(1H-indol-3-yl)-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(thiophene-2-carbonyl)piperidine
N-(pyridin-3-ylmethyl)-1-[1-(1,2,3,4-tetrahydronaphthalen-2-yl)piperidin-4-yl]piperidine-4-carboxamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]piperidine-1-carboxamide
2-(3-chloro-2,6-difluorophenyl)-1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]ethan-1-one
(1H-imidazol-2-ylmethyl)(3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl)amine
1-{3-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(3S,4R)-4-(4-methylphenyl)-1-(6-oxo-1,6-dihydropyridine-3-carbonyl)pyrrolidin-3-yl]cyclopropanecarboxamide
4-(ethanesulfonyl)-2-[2-(oxolan-3-yl)-1H-imidazol-1-yl]phenol
N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-4-(2-methoxyethyl)piperazine
7-(2-methoxyethyl)-2-{2-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2,7-diazaspiro[4.5]decan-6-one
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[(4-methyl-1,3-thiazol-2-yl)methyl]benzamide