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N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-methoxy-N-methyl-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazole
2-(pyridin-3-yl)-2-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}ethan-1-ol
1-[(3R,4S)-3-[(4-ethyl-5-methylpyrimidin-2-yl)amino]-4-(propan-2-yl)pyrrolidine-1-carbonyl]cyclopropane-1-carboxamide
1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(propan-2-yloxy)propan-1-one
2-ethoxy-6-[({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]phenol
2-[1-(5-chloro-3-phenyl-1H-indol-2-yl)-N-methylformamido]-N-methylacetamide
8-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(1-ethyl-1H-pyrazol-4-yl)methyl]amine
methyl 5-[(4-hydroxybutan-2-yl)amino]-3-(oxolane-2-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)acetamide
2-(4-{[4-(2-methylpropyl)phenyl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
N-ethyl-1-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidine-3-carboxamide
6-ethyl-4-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-2H-chromen-2-one
2-ethyl-1-(propan-2-yl)-4-[6-(pyridin-4-yl)pyridine-3-carbonyl]piperazine
5-({4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}methyl)-2-methoxybenzoic acid
2-methyl-6-(1-{1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-yl)pyrimidin-4-ol
N-benzyl-2-[2-(2-methoxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]acetamide
4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-(prop-2-en-1-yl)benzamide
3-[({[5-(4-chlorophenyl)furan-2-yl]methyl}amino)methyl]-5-methanesulfonamido-N-(propan-2-yl)benzamide
N-{[7-chloro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]acetamide
1-cycloheptyl-4-{[(1-methyl-1H-imidazol-2-yl)methyl]amino}pyrrolidin-2-one
1-[2-(8-methoxyquinolin-5-yl)pyrimidin-4-yl]pyrrolidin-3-ol
3-fluoro-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidine-4-carboxylic acid
2-[1-(3-phenylpropyl)-4-(1H-pyrazole-3-carbonyl)piperazin-2-yl]ethan-1-ol
{2-[4-(8-chloroquinoline-2-carbonyl)morpholin-2-yl]ethyl}dimethylamine
methyl (2S,4S,5R)-1,2-dimethyl-4-(1,2-oxazinane-2-carbonyl)-5-phenylpyrrolidine-2-carboxylate
3-methyl-1-{7-[(4-methylpiperazin-1-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}butan-1-one
1-methyl-N-[(5-methylpyrazin-2-yl)methyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(5-ethylpyridin-2-yl)methyl]-N,1,3-trimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-cyclohexyl-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]piperidine-4-carboxamide
methyl 3-(4-{[4-(piperidine-1-carbonyl)piperidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoate
3-methyl-N-[(3-propyl-1,2-oxazol-5-yl)methyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
4-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(2-oxoimidazolidin-1-yl)-N-propylbenzamide
3-{[3-(2-hydroxyethyl)-4-(thiophen-3-ylmethyl)piperazin-1-yl]methyl}-6-methyl-4H-chromen-4-one
N-[2-(3-phenyl-1H-1,2,4-triazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide
1-[4-(ethylcarbamoyl)pyridin-2-yl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
4-(3-ethyl-1H-indole-2-carbonyl)-1-(4-methoxyphenyl)piperazin-2-one
4-(benzyloxy)-N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]butanamide
1-[2-(3-fluorophenyl)ethyl]-6-oxo-N-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-3-carboxamide
(3R,9aR)-3-(hydroxymethyl)-8-(3-methylbutyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}naphthalen-2-ol
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-5-methoxyfuran-2-carboxamide
(7R,9aR)-N-(3-fluorophenyl)-7-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
1-{6-[3-(ethylsulfanyl)phenyl]pyridin-2-yl}ethan-1-ol
(2S)-N-[2-chloro-5-(piperidine-1-carbonyl)phenyl]-2-(hydroxymethyl)pyrrolidine-1-carboxamide
N-[(2-fluorophenyl)methyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3aR,6aS)-2-(cyclopropylmethyl)-5-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid