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7-(2,3-dihydro-1,4-benzodioxine-5-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
methyl 4-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}amino)benzoate
N-[(5-methoxy-1H-indol-2-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
N-[(3,4-difluorophenyl)methyl]-3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)propanamide
2-[3-(4-methoxyphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-2-azabicyclo[2.2.1]heptane
3-oxo-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
(2S,4R)-4-amino-1-[(5-cyclohexylthiophen-2-yl)methyl]-N-methylpyrrolidine-2-carboxamide
4-methyl-3-oxo-N-(4-{[2-(pyridin-2-yl)ethyl]sulfanyl}phenyl)piperazine-1-carboxamide
N-methyl-N-{2-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}benzenesulfonamide
1-(2-fluorophenyl)-N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}cyclopropane-1-carboxamide
(4aR,7aS)-4-[(3-methoxyphenyl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-{3-[cyclopentyl(methyl)amino]propyl}-2-(1H-imidazol-2-yl)benzamide
1-[2-(2,2-dimethyloxan-4-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]piperidine-3-carboxamide
3-[2-(2-hydroxyphenyl)acetyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-amine
1-benzyl-N3-[(1R)-1-(3-methoxyphenyl)ethyl]-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-methyl-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-(6-methoxypyrimidin-4-yl)phenol
7-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
N-[(1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)methyl]pyridine-3-carboxamide
1-benzyl-N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-1H-pyrazole-4-carboxamide
3-{5-[4-methyl-3-(1H-pyrrol-1-yl)benzoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-(1,2-diphenylethyl)-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
N-[1-(7-{[3-(2-hydroxyethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-3-phenylpropanamide
2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-propylacetamide
4-(2,2-diphenylethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-[(6-methoxypyrimidin-4-yl)amino]-7-methyl-2,3-dihydro-1H-indol-2-one
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-7-(2-methoxyacetamido)-1-methyl-2-(pyridin-3-yl)-1H-1,3-benzodiazole-5-carboxamide
2-[(2-fluorophenyl)amino]-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine
4-(8-fluoro-4-oxo-1,4-dihydroquinoline-2-carbonyl)-1λ6-thiomorpholine-1,1-dione
3-[3-methyl-5-(pyrrolidin-1-ylmethyl)phenoxy]-6-phenylpyridazine
8-fluoro-2-[3-(pyridine-3-carbonyl)piperidine-1-carbonyl]quinoline
2-amino-4-(3-methylthiophen-2-yl)-6-(pyridin-3-yl)pyridine-3-carbonitrile
2-[4-(3-methylfuran-2-carbonyl)-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(5-methylfuran-2-yl)methyl]pyrimidin-2-amine
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}urea
1-cyclopentyl-N-(furan-3-ylmethyl)-5-oxopyrrolidine-3-carboxamide
2-[3-(1,3-dimethyl-1H-pyrazol-4-yl)-1H-pyrazol-1-yl]-N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)acetamide
3-butyl-5-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidine
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]({[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl})methylamine
(2R,3R)-3-[(3-methoxypropyl)(methyl)amino]-1'-(3-methylbut-2-en-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-ethylpyrimidin-2-amine
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
5-chloro-6-oxo-N-[1-(2-phenylethyl)piperidin-3-yl]-1,6-dihydropyridine-3-carboxamide
2-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2-oxoacetamide
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-4-(1H-pyrazol-4-yl)butanamide
4-(5-methoxy-3-methyl-1H-indole-2-carbonyl)piperazine-2-carboxylic acid
N-(2-cyclopentyl-2-phenylethyl)-2-(pyridin-3-yl)acetamide