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(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(pyridin-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(2-phenylethyl)-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
N-[2-(diethylamino)ethyl]-N-ethyl-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-[2-(5-methylfuran-2-yl)ethyl]acetamide
methyl 3-[(3-hydroxyphenyl)methyl]-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(2,3-dimethoxybenzoyl)-3-(1-methyl-1H-imidazol-2-yl)piperidine
5-(5-methoxyfuran-2-yl)-3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
{4-[(5-chloro-3-methoxy-2-propoxyphenyl)methyl]-1-methylpiperazin-2-yl}methanol
1-(1'-{[2-(propylamino)pyrimidin-5-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
N3-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-1-cyclopentyl-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[(4-fluorophenyl)methyl]-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
N-[(1S,2R)-2-(hydroxymethyl)cyclopentyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
8-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
(1R,5R)-N,N-dimethyl-6-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(4aR,7aS)-1-{2-[(furan-3-ylmethyl)(methyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{6-hydroxy-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-1-yl}-2,2-bis(hydroxymethyl)butan-1-one
6-[2-(aminomethyl)-5-fluoro-2,3-dihydro-1-benzofuran-7-yl]-2H-1,3-benzodioxole-5-carboxamide
2-benzyl-N-[2-(2-methoxyphenyl)ethyl]-1,3-thiazole-4-carboxamide
1-methyl-4-({5-[2-(1H-1,2,3,4-tetrazol-1-yl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl}methyl)piperidine
N-[1-(2-chlorophenyl)cyclopropyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)but-2-enamide
[(5-{1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[2-(2-fluorophenoxy)ethyl]acetamide
N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
5-(2,4-difluorophenoxymethyl)-N-methyl-N-(2-methylprop-2-en-1-yl)-1,2-oxazole-3-carboxamide
2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylacetamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2-oxo-2-(piperidin-1-yl)acetamide
(2S,4S)-4-amino-1-(2,1,3-benzothiadiazole-4-sulfonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-{5-[(3-acetamidopyrrolidin-1-yl)methyl]-1,2,4-oxadiazol-3-yl}benzoic acid
(2S)-2-amino-1-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-(1H-imidazol-4-yl)propan-1-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(2,6-dimethoxyphenyl)methyl]benzamide
3-{[2-(piperidin-1-yl)-2,3-dihydro-1H-inden-2-yl]formamido}propanamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetamide
8-methyl-3-[2-(trifluoromethyl)morpholine-4-carbonyl]-1,4-dihydroquinolin-4-one
2,2-difluoro-N-{[1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)pyrrolidin-3-yl]methyl}acetamide
N-{1-[7-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}pyridine-3-carboxamide
3-(3-fluorophenyl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
(2S)-3-(1H-indol-3-yl)-2-[(5-methanesulfonyl-2-methylpyrimidin-4-yl)amino]propan-1-ol
{5-[1-(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methanol
1-(isoquinolin-5-ylmethyl)-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-4-carboxamide
2-methyl-4-(5-{[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}thiophen-2-yl)but-3-yn-2-ol
2-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propane-1,3-diol
2-[1-(3-methylbut-2-en-1-yl)-4-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperazin-2-yl]ethan-1-ol
4-methoxy-6-[4-(pyridin-3-yloxy)piperidin-1-yl]pyrimidine
6-{[4-(oxan-4-yl)piperazin-1-yl]methyl}naphthalen-2-ol
1-(2-methoxyethyl)-6-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]piperidine-3-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-4-(pyridin-2-yl)pyrimidin-2-amine
4-[(3,3-diphenylpiperidin-1-yl)methyl]-N-methylbenzamide
(1S,5R)-3-(3-fluoropyridin-4-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(1H-imidazol-2-ylmethyl)-N-[2-(4-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide