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N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-4-(piperidin-3-yl)benzamide
6-methyl-N,N-bis(1,3-oxazol-4-ylmethyl)imidazo[2,1-b][1,3]thiazole-5-carboxamide
3-[(4-hydroxy-6-methylpyrimidin-2-yl)methyl]-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
4-{3-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]propanamido}benzamide
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(pyridazine-3-carbonyl)piperidine-4-carboxylic acid
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1-methyl-1H-indole-6-carboxamide
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-phenylpiperidin-4-ol
3-{1-[6-amino-2-(morpholin-4-yl)pyrimidin-4-yl]piperidin-3-yl}-N,N-dimethylpropanamide
1-(2-methoxyacetyl)-N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]piperidine-4-carboxamide
4-(dimethylamino)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
5-propyl-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}pyrazolo[1,5-a]pyrimidin-7-amine
5-(1H-imidazol-1-ylmethyl)-3-(2-methoxyethyl)-1-[(3-methylphenyl)methyl]-1H-1,2,4-triazole
[(3S,7S)-5-(4-chlorobenzoyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-trien-3-yl]methanol
1-({5-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]furan-2-yl}methyl)-4-methylpiperidine
(1R,2S)-N-methyl-2-[1-phenyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]cyclohexane-1-carboxamide
3-(azepane-1-carbonyl)-N-(3-ethoxypropyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-methyl-2-oxo-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-oxaspiro[4.5]decane-4-carboxamide
1-(2-methoxyethyl)-N3-[(4-methoxyphenyl)methyl]-4-oxo-N5-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-(but-3-enoyl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-({[1-(1-methyl-1H-imidazole-2-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
2-(dimethylamino)-2-(4-methylphenyl)-N-{3-[(pyridin-3-yl)amino]propyl}acetamide
5-[4-(aminomethyl)piperidin-1-yl]-2-[2-(1-methylpiperidin-2-yl)ethyl]-2,3-dihydropyridazin-3-one
3-methyl-1-[3-(4-methylphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine
(2E)-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)-3-(thiophen-2-yl)prop-2-enamide
2-(3-cyano-2-methoxypyridin-4-yl)-6-methoxy-N,N-bis(propan-2-yl)benzamide
dimethyl(3-{2-[1-(6-methylpyridine-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
4-(1-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}piperidine-4-carbonyl)morpholine
2-{3-[(4-fluoropiperidin-1-yl)methyl]phenoxy}acetamide
{3-[(3-methoxyphenyl)methyl]-1-(3-phenylprop-2-yn-1-yl)piperidin-3-yl}methanol
N-[(4-acetamidophenyl)methyl]-2-[(1H-imidazol-2-ylmethyl)amino]acetamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-5-fluoro-N-(2-hydroxyethyl)-1,3-dimethyl-1H-indole-2-carboxamide
3-{[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,2-benzoxazole
2-(4-acetylphenoxy)-1-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]ethan-1-one
ethyl 1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-3-carboxylate
N-ethyl-2-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)acetamide
N-methyl-5-(phenoxymethyl)-N-(1-phenylpropyl)-1H-pyrazole-3-carboxamide
5-cyclobutanecarbonyl-1'-[(4-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-cyclopropyl-2-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methoxy}benzamide
(4aS,7aR)-1-(8-hydroxyquinoline-7-carbonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[3-(4-{[3-(furan-2-yl)-3-phenylpropyl]amino}piperidin-1-yl)phenyl]cyclopropanecarboxamide
(1S,5R)-6-(2-methoxyethyl)-3-(5-methyl-1,3-benzoxazol-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(4-{[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]methyl}phenyl)ethan-1-one
2-[3-({methyl[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]acetamide
3-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridin-2-ol
8-methoxy-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
4-{1-[(2-chloro-3,4-dimethoxyphenyl)methyl]piperidin-3-yl}-5-(4-fluorophenyl)-2-methylpyrimidine
1-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-(prop-2-en-1-yl)urea
1-[(2E)-3-(3,4-difluorophenyl)prop-2-enoyl]-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one